SCHEMBL2664841

SCHEMBL2664841

O=C(Nc1nccs1)C(CC1CCCC1)c1ccc(-c2cncnc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GCK P35557 10/20 0.68
FFAR2 O15552 5/20 0.66
KCNH2 Q12809 1/20 0.59
EPHX2 P34913 1/20 0.48
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2647122 0.91 GCK (0.71) GCKFFAR2KCNH2EPHX2CYP1A2
SCHEMBL2647322 0.90 GCK (0.66) GCKFFAR2KCNH2EPHX2CYP1A2
SCHEMBL2647740 0.89 GCK (0.71) GCKFFAR2KCNH2EPHX2CYP1A2
SCHEMBL2647924 0.89 GCK (0.71) GCKFFAR2KCNH2EPHX2CYP1A2
SCHEMBL2650901 0.87 GCK (0.65) GCKFFAR2KCNH2EPHX2CYP1A2
SCHEMBL2654951 0.86 GCK (0.74) GCKFFAR2KCNH2EPHX2CYP1A2
SCHEMBL2644739 0.85 GCK (0.76) GCKFFAR2KCNH2EPHX2CYP1A2
SCHEMBL2645871 0.84 GCK (0.74) GCKFFAR2KCNH2EPHX2CYP1A2
SCHEMBL2645293 0.84 GCK (0.74) GCKFFAR2KCNH2EPHX2CYP1A2
SCHEMBL2646757 0.84 FFAR2 (0.91) GCKFFAR2KCNH2EPHX2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001083465-A2 ALKYNYL PHENYL HETEROAROMATIC GLUCOKINASE ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2001-11-08 WO disclosed