SCHEMBL26655331

SCHEMBL26655331

CNc1nc(Nc2ccc(C(=O)N3CCN(Cc4ccc(CBr)cc4)CC3)cc2OC)ncc1Cl

nearest known ligand 0.75

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 20/20 0.75
MAP3K9 P80192 1/20 0.71
MKNK2 Q9HBH9 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30680126 1.00 LRRK2 (0.75) LRRK2MAP3K9MKNK2
SCHEMBL26655184 0.94 LRRK2 (0.70) LRRK2MAP3K9MKNK2
SCHEMBL30680150 0.94 LRRK2 (0.70) LRRK2MAP3K9MKNK2
SCHEMBL30680139 0.89 LRRK2 (0.78) LRRK2
SCHEMBL26655477 0.89 LRRK2 (0.78) LRRK2
SCHEMBL14556200 0.88 LRRK2 (0.82) LRRK2MAP3K9MKNK2
SCHEMBL26655374 0.88 LRRK2 (0.76) LRRK2MAP3K9MKNK2
SCHEMBL30680138 0.88 LRRK2 (0.76) LRRK2MAP3K9MKNK2
SCHEMBL14860253 0.87 LRRK2 (0.79) LRRK2MAP3K9MKNK2
SCHEMBL30636053 0.87 LRRK2 (0.79) LRRK2MAP3K9MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260001875-A1 AMINOPYRIMIDINYL DERIVATIVES FOR THE TREATMENT OF PARKINSON'S DISEASE UNIV DUNDEE (GB) 2026-01-01 US disclosed
WO-2023218187-A1 AMINOPYRIMIDINYL DERIVATIVES FOR THE TREAMENT OF PARKINSON'S DISEASE UNIVERSITY OF DUNDEE (GB) 2023-11-16 WO disclosed
WO-2023218187-A1 AMINOPYRIMIDINYL DERIVATIVES FOR THE TREAMENT OF PARKINSON'S DISEASE UNIVERSITY OF DUNDEE (GB) 2023-11-16 WO disclosed
EP-4276097-A1 AMINOPYRIMIDINYL DERIVATIVES FOR THE TREAMENT OF PARKINSON'S DISEASE University Of Dundee (GB) 2023-11-15 EP disclosed
EP-4276097-A1 AMINOPYRIMIDINYL DERIVATIVES FOR THE TREAMENT OF PARKINSON'S DISEASE University Of Dundee (GB) 2023-11-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260001875-A1 AMINOPYRIMIDINYL DERIVATIVES FOR THE TREATMENT OF PARKINSON'S DISEASE LRRK2, XIAP, PARK7 LRRK2 1/4885MAP3K9 1699/4885MKNK2 266/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.