SCHEMBL2666752

SCHEMBL2666752

CS(=O)(=O)c1ccc(/C(=N\OC2CCCC2)C(=O)Nc2ncc(C(F)(F)F)s2)cc1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GCK P35557 11/20 0.43
KCNH2 Q12809 4/20 0.42
CDK2 P24941 1/20 0.38
KDR P35968 1/20 0.38
FFAR2 O15552 2/20 0.38
PTGS1 P23219 2/20 0.36
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10230994 0.88 GCK (0.47) GCKKCNH2
SCHEMBL2666841 0.87 GCK (0.46) GCKKCNH2KMT2A
SCHEMBL10230984 0.86 GCK (0.56) GCKKCNH2
SCHEMBL10231004 0.86 GCK (0.45) GCKKCNH2KMT2A
SCHEMBL9072364 0.85 GCK (0.45) GCKKCNH2CDK2KDRFFAR2
SCHEMBL10230964 0.85 GCK (0.46) GCKKCNH2KMT2A
SCHEMBL2666751 0.85 GCK (0.44) GCKKCNH2FFAR2KMT2A
SCHEMBL10230961 0.85 GCK (0.44) GCKKCNH2FFAR2KMT2A
SCHEMBL10230968 0.85 GCK (0.46) GCKKCNH2KMT2A
SCHEMBL2666983 0.84 GCK (0.43) GCKKCNH2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119626-B2 Oxime derivative and preparations thereof MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-02-21 US disclosed
US-8119626-B2 Oxime derivative and preparations thereof MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-02-21 US disclosed
US-20090291936-A1 OXIME DERIVATIVE AND PREPARATIONS THEREOF SUGAWARA KAZUTOSHI 2009-11-26 US disclosed
US-20090291936-A1 OXIME DERIVATIVE AND PREPARATIONS THEREOF SUGAWARA KAZUTOSHI 2009-11-26 US disclosed
US-7514439-B2 Oxime derivative and preparations thereof MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-04-07 US disclosed
US-7514439-B2 Oxime derivative and preparations thereof MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-04-07 US disclosed
US-20080132479-A1 Oxime Derivative and Preparations Thereof MITSUBISHI TANABE PHARMA CORPORATION (JP) 2008-06-05 US disclosed
US-20080132479-A1 Oxime Derivative and Preparations Thereof MITSUBISHI TANABE PHARMA CORPORATION (JP) 2008-06-05 US disclosed
WO-2007007886-A1 AN OXIME DERIVATIVE AND PREPARATIONS THEREOF MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-01-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080132479-A1 Oxime Derivative and Preparations Thereof GCK, KHK, GCKR GCK 1/4885KCNH2 291/4885CDK2 342/4885
US-20090291936-A1 OXIME DERIVATIVE AND PREPARATIONS THEREOF GCK, KHK, GCKR GCK 1/4885KCNH2 291/4885CDK2 342/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.