SCHEMBL2667720

SCHEMBL2667720

COC(=O)Cc1ccc(NC(=O)c2cc(Oc3ccc(NC(=O)c4ccccc4)cc3)nc(OC(C)C)c2)nc1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GCK P35557 12/20 0.49
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
LOX P28300 2/20 0.44
LOXL2 Q9Y4K0 2/20 0.44
POLB P06746 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2667760 0.93 GCK (0.44) GCKMEN1KMT2ANPC1RAB9A
SCHEMBL2667809 0.93 GCK (0.53) GCKMEN1KMT2A
SCHEMBL2667776 0.91 GCK (0.51) GCKMEN1KMT2A
SCHEMBL9070996 0.90 GCK (0.50) GCK
SCHEMBL2667360 0.89 LMNA (0.45) GCK
SCHEMBL2667442 0.87 GCK (0.57) GCK
SCHEMBL2667620 0.87 GCK (0.46) GCK
SCHEMBL9071038 0.86 GCK (0.48) GCK
SCHEMBL2667562 0.86 GCK (0.47) GCK
SCHEMBL2667633 0.86 GCK (0.53) GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009083553-A1 AZINE COMPOUNDS AS GLUCOKINASE ACTIVATORS RHEOSCIENCE A/S (DK) 2009-07-09 WO disclosed