SCHEMBL26684381

SCHEMBL26684381

COC(=O)c1cn(C(C(=O)O)C(C)C)nn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.40
CA1 P00915 4/20 0.40
CA2 P00918 4/20 0.40
CA9 Q16790 4/20 0.40
MGAM O43451 1/20 0.39
GAA P10253 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
NOTUM Q6P988 4/20 0.39
LGALS3 P17931 1/20 0.36
DPP4 P27487 2/20 0.34
CA3 P07451 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
CA5A P35218 1/20 0.33
CA7 P43166 1/20 0.33
CA13 Q8N1Q1 1/20 0.33
CA14 Q9ULX7 1/20 0.33
CA5B Q9Y2D0 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26683331 1.00 CA12 (0.40) CA12CA1CA2CA9MGAM
SCHEMBL1155520 0.84 CA12 (0.42) CA12CA1CA2CA9MGAM
SCHEMBL26684401 0.84 HTT (0.39) LGALS3ALDH1A1LMNAPTPN1CDC25B
SCHEMBL26684394 0.84 HTT (0.39) LGALS3ALDH1A1LMNAPTPN1CDC25B
SCHEMBL12862751 0.83 CA12 (0.43) CA12CA1CA2CA9MGAM
SCHEMBL14262390 0.82 CA12 (0.44) CA12CA1CA2CA9MGAM
SCHEMBL11983464 0.78 CA12 (0.42) CA12CA1CA2CA9MGAM
SCHEMBL31124085 0.78 CA12 (0.45) CA12CA1CA2CA9MGAM
SCHEMBL31605659 0.76 LGALS3 (0.35) CA12CA1CA2CA9LGALS3
SCHEMBL909222 0.72 HTT (0.44) CA12CA1CA2CA9MGAM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023220237-A1 BENZOTHIAZOLE COMPOUNDS AS VHL LIGANDS GENENTECH, INC. (US) 2023-11-16 WO disclosed