SCHEMBL26697299

SCHEMBL26697299

COc1cc2c(Oc3ccc(NC(=O)Nc4cc(C)on4)c(Cl)c3)ncnc2cc1O

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 15/20 0.70
FLT1 P17948 4/20 0.70
FLT4 P35916 4/20 0.70
PDGFRA P16234 3/20 0.68
EPHB2 P29323 2/20 0.68
KIT P10721 2/20 0.68
RIPK2 O43353 1/20 0.68
STK10 O94804 1/20 0.68
ABL1 P00519 1/20 0.68
LCK P06239 1/20 0.68
LYN P07948 1/20 0.68
RET P07949 1/20 0.68
MET P08581 1/20 0.68
PDGFRB P09619 1/20 0.68
BCR P11274 1/20 0.68
FGFR1 P11362 1/20 0.68
SRC P12931 1/20 0.68
MAPK3 P27361 1/20 0.68
HTR2A P28223 1/20 0.68
MAPK1 P28482 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5653965 0.94 KDR (0.78) KDRFLT1FLT4PDGFRAEPHB2
SCHEMBL24520229 0.91 KDR (0.74) KDRFLT1FLT4PDGFRAEPHB2
SCHEMBL15962801 0.88 KDR (0.82) KDRFLT1FLT4PDGFRAEPHB2
SCHEMBL24520230 0.88 KDR (0.82) KDRFLT1FLT4PDGFRAEPHB2
SCHEMBL15962810 0.87 KDR (0.89) KDRFLT1FLT4PDGFRAEPHB2
SCHEMBL26697261 0.87 KDR (0.73) KDRFLT1FLT4PDGFRAEPHB2
SCHEMBL15962835 0.86 KDR (0.79) KDRFLT1FLT4PDGFRAEPHB2
SCHEMBL26894876 0.86 KDR (0.68) KDRFLT1FLT4PDGFRAKIT
SCHEMBL5206338 0.86 KDR (0.68) KDRFLT1FLT4PDGFRAKIT
SCHEMBL26697206 0.85 KDR (0.70) KDRFLT1FLT4PDGFRAKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114920703-B Quinazoline derivative and preparation method and application thereof 天津济坤医药科技有限公司 2024-01-09 CN disclosed
WO-2023226323-A1 QUINAZOLINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 天津济坤医药科技有限公司 2023-11-30 WO disclosed
WO-2023226323-A1 QUINAZOLINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 天津济坤医药科技有限公司 2023-11-30 WO disclosed
CN-114920703-A Quinazoline derivative and preparation method and application thereof 天津济坤医药科技有限公司 2022-08-19 CN disclosed