SCHEMBL26697304

SCHEMBL26697304

O=C(Nc1cccc(C(F)(F)F)c1)Nc1ccc(O)cc1Cl

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.74
TRPV1 Q8NER1 3/20 0.69
NTRK1 P04629 1/20 0.66
CDK19 Q9BWU1 1/20 0.66
MEN1 O00255 3/20 0.62
KMT2A Q03164 3/20 0.62
MAPT P10636 2/20 0.62
HTT P42858 1/20 0.62
RAB9A P51151 1/20 0.62
GRIK1 P39086 7/20 0.62
BAZ1A Q9NRL2 1/20 0.58
ALDH1A1 P00352 3/20 0.57
CYP1A2 P05177 1/20 0.57
POLB P06746 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
XBP1 P17861 1/20 0.57
CYP2C19 P33261 1/20 0.57
RXFP1 Q9HBX9 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14459439 0.88 KDR (0.76) KDRTRPV1NTRK1CDK19MEN1
SCHEMBL1463622 0.87 TRPV1 (0.70) KDRTRPV1NTRK1CDK19MEN1
SCHEMBL10991763 0.85 KDR (1.00) KDRTRPV1NTRK1CDK19MEN1
SCHEMBL26697260 0.85 CA12 (0.64) KDRTRPV1MEN1KMT2AMAPT
SCHEMBL1463509 0.85 GRIK1 (0.77) KDRTRPV1NTRK1CDK19MEN1
SCHEMBL3676521 0.85 TRPV1 (0.67) KDRTRPV1NTRK1CDK19MEN1
SCHEMBL1463407 0.84 NTRK1 (0.77) KDRTRPV1NTRK1CDK19MEN1
SCHEMBL5594672 0.84 KDR (0.69) KDRTRPV1NTRK1CDK19MEN1
SCHEMBL26697226 0.83 TRPV1 (0.64) KDRTRPV1MEN1KMT2AMAPT
SCHEMBL6370948 0.82 TRPV1 (0.64) KDRTRPV1NTRK1CDK19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114920703-B Quinazoline derivative and preparation method and application thereof 天津济坤医药科技有限公司 2024-01-09 CN disclosed
WO-2023226323-A1 QUINAZOLINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 天津济坤医药科技有限公司 2023-11-30 WO disclosed
CN-114920703-A Quinazoline derivative and preparation method and application thereof 天津济坤医药科技有限公司 2022-08-19 CN disclosed