SCHEMBL26697226

SCHEMBL26697226

O=C(Nc1cccc(F)c1)Nc1ccc(O)cc1Cl

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 6/20 0.64
RAB9A P51151 5/20 0.62
MEN1 O00255 4/20 0.62
KMT2A Q03164 4/20 0.62
GRIK1 P39086 1/20 0.57
MAPT P10636 4/20 0.54
NPC1 O15118 3/20 0.52
SMN1; SMN2 Q16637 2/20 0.51
MTOR P42345 1/20 0.51
TAAR1 Q96RJ0 1/20 0.51
GAA P10253 1/20 0.51
PTGER3 P43115 1/20 0.51
HTT P42858 1/20 0.50
ATM Q13315 1/20 0.50
KDR P35968 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21751042 0.86 MEN1 (0.62) TRPV1RAB9AMEN1KMT2AGRIK1
SCHEMBL4554472 0.84 KDR (0.68) TRPV1RAB9AMEN1KMT2AGRIK1
SCHEMBL21750906 0.84 RAB9A (0.56) TRPV1RAB9AMEN1KMT2AGRIK1
SCHEMBL29757932 0.84 RAB9A (0.56) TRPV1RAB9AMEN1KMT2AGRIK1
SCHEMBL21750979 0.84 MAOA (0.61) TRPV1RAB9AMEN1KMT2AGRIK1
SCHEMBL29757943 0.84 MAOA (0.61) TRPV1RAB9AMEN1KMT2AGRIK1
SCHEMBL26697304 0.83 KDR (0.74) TRPV1RAB9AMEN1KMT2AGRIK1
SCHEMBL24272323 0.81 MTOR (0.69) TRPV1RAB9AMEN1KMT2AMAPT
SCHEMBL30851500 0.80 RAB9A (0.79) RAB9AMEN1KMT2AMAPTNPC1
SCHEMBL27193042 0.80 RAB9A (0.79) RAB9AMEN1KMT2AMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114920703-B Quinazoline derivative and preparation method and application thereof 天津济坤医药科技有限公司 2024-01-09 CN disclosed
WO-2023226323-A1 QUINAZOLINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 天津济坤医药科技有限公司 2023-11-30 WO disclosed
WO-2023226323-A1 QUINAZOLINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 天津济坤医药科技有限公司 2023-11-30 WO disclosed
CN-114920703-A Quinazoline derivative and preparation method and application thereof 天津济坤医药科技有限公司 2022-08-19 CN disclosed