SCHEMBL2677484

SCHEMBL2677484

NC(=O)c1cc(CN2CCOCC2)ccc1C(=O)Nc1n[nH]c2c1CN(S(=O)(=O)c1cc(F)cc(F)c1)CC2

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 4/20 0.55
INSR P06213 2/20 0.42
ALK Q9UM73 2/20 0.42
NTRK1 P04629 2/20 0.39
NTRK3 Q16288 2/20 0.39
NTRK2 Q16620 2/20 0.39
SMN1; SMN2 Q16637 4/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
MAPK1 P28482 2/20 0.37
ALDH1A1 P00352 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
LMNA P02545 2/20 0.37
HTT P42858 1/20 0.37
NPC1 O15118 4/20 0.36
RAB9A P51151 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2678322 0.93 IGF1R (0.55) IGF1RINSRALKNTRK1SMN1; SMN2
SCHEMBL2677489 0.92 IGF1R (0.56) IGF1RINSRALKNTRK1NTRK3
SCHEMBL2678132 0.87 IGF1R (0.65) IGF1RINSRALKNTRK1NTRK3
SCHEMBL1889800 0.87 INSR (0.57) IGF1RINSRALKNTRK1NTRK3
SCHEMBL2678223 0.87 NTRK1 (0.46) IGF1RINSRALKNTRK1NTRK3
SCHEMBL2452437 0.87 IGF1R (0.52) IGF1RINSRALKNTRK1NTRK3
SCHEMBL1886125 0.85 IGF1R (0.56) IGF1RINSRALKNTRK1NTRK3
SCHEMBL1882045 0.85 IGF1R (0.69) IGF1RINSRALKNTRK1NTRK3
SCHEMBL2678327 0.85 IGF1R (0.56) IGF1RINSRALKNTRK1TP53
SCHEMBL1891292 0.85 IGF1R (0.50) IGF1RINSRALKNTRK1NTRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8173659-B2 Substituted pyrazolo[4,3-C]pyridine derivatives active as kinase inhibitors NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2012-05-08 US disclosed
US-20090023745-A1 Substituted Pyrazolo[4,3-c]Pyridine Derivatives Active as Kinase Inhibitors NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2009-01-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090023745-A1 Substituted Pyrazolo[4,3-c]Pyridine Derivatives Active as Kinase Inhibitors MAP3K3, MAP3K1, MAP3K19 IGF1R 760/4885INSR 922/4885ALK 517/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.