SCHEMBL2690752

SCHEMBL2690752

CC(N)c1ccc(OCCF)nc1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
APP P05067 5/20 0.39
MAPT P10636 1/20 0.39
SNCA P37840 1/20 0.39
ACACB O00763 4/20 0.35
ADRB2 P07550 1/20 0.33
FFAR1 O14842 3/20 0.32
PDE2A O00408 1/20 0.32
PTGES O14684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14480145 0.87 PIK3CD (0.41) MAPTACACBADRB2FFAR1
SCHEMBL18266151 0.87 PIK3CD (0.41) MAPTACACBADRB2FFAR1
SCHEMBL19398567 0.86 APP (0.40) APPMAPTSNCAACACBFFAR1
SCHEMBL18266621 0.85 ACACB (0.47) MAPTACACB
SCHEMBL14480054 0.83 PIK3CD (0.42) ACACBADRB2FFAR1PTGES
SCHEMBL17002596 0.83 APP (0.39) APPMAPTSNCAACACBFFAR1
SCHEMBL19764493 0.83 PIK3CD (0.42) ACACBADRB2FFAR1PTGES
SCHEMBL4550384 0.83 EPHX2 (0.41) ACACBPDE2A
Hydrochloric Acid SCHEMBL2714794 0.81 EPHX2 (0.41) ACACBPDE2A
SCHEMBL14480391 0.81 MAPT (0.46) MAPTACACBADRB2FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100286202-A1 New Compounds ASTRAZENECA AB (SE) 2010-11-11 US claimed
EP-1966156-A2 NEW COMPOUNDS III AstraZeneca AB (SE) 2008-09-10 EP claimed
US-20080171770-A1 Compounds ASTRAZENECA AB (SE) 2008-07-17 US claimed
WO-2007073303-A2 NOVEL BENZIMIDAZOLE DERIVATIVES AS VANILLOID RECEPTOR 1 (VRL) INHIBITORS ASTRAZENECA AB (SE) 2007-06-28 WO claimed
EP-3632899-A1 ARYL SUBSTITUTED CARBOXAMIDE DERIVATIVES AS CALCIUM OR SODIUM CHANNEL BLOCKERS RaQualia Pharma Inc. (JP) 2020-04-08 EP disclosed
US-8168668-B2 Compounds ASTRAZENECA AB (SE) 2012-05-01 US disclosed
EP-1966156-B1 NEW COMPOUNDS III ASTRAZENECA AB (SE) 2011-12-21 EP disclosed
US-8008487-B2 Substituted thieno[2,3-D]pyrimidines as fungicides DOW AGROSCIENCES LLC (US) 2011-08-30 US disclosed
US-8008487-B2 Substituted thieno[2,3-D]pyrimidines as fungicides DOW AGROSCIENCES LLC (US) 2011-08-30 US disclosed
US-20100286202-A1 New Compounds ASTRAZENECA AB (SE) 2010-11-11 US disclosed
US-7618993-B2 Compounds ASTRAZENECA AB (SE) 2009-11-17 US disclosed
EP-1966156-A2 NEW COMPOUNDS III AstraZeneca AB (SE) 2008-09-10 EP disclosed
US-20080171770-A1 Compounds ASTRAZENECA AB (SE) 2008-07-17 US disclosed
WO-2007073303-A2 NOVEL BENZIMIDAZOLE DERIVATIVES AS VANILLOID RECEPTOR 1 (VRL) INHIBITORS ASTRAZENECA AB (SE) 2007-06-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100286202-A1 New Compounds REN, PCSK9, FURIN APP 372/4885MAPT 67/4885SNCA 1514/4885
US-20080171770-A1 Compounds REN, PCSK9, SLC10A1 APP 373/4885MAPT 102/4885SNCA 805/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.