SCHEMBL26940527

SCHEMBL26940527

COC(=O)C1CC(Oc2cccc(Br)c2)CN1C(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 1/20 0.46
NR1H2 P55055 1/20 0.44
NR1H3 Q13133 1/20 0.44
MCL1 Q07820 11/20 0.44
KCNH2 Q12809 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
USP30 Q70CQ3 1/20 0.41
PTPN1 P18031 1/20 0.40
BCL2 P10415 1/20 0.39
BCL2L1 Q07817 1/20 0.39
UCHL1 P09936 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
CYP1A2 P05177 1/20 0.38
POLB P06746 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26940536 1.00 P2RX3 (0.46) P2RX3NR1H2NR1H3MCL1KCNH2
SCHEMBL31336371 1.00 P2RX3 (0.46) P2RX3NR1H2NR1H3MCL1KCNH2
SCHEMBL3862645 0.89 P2RX3 (0.47) P2RX3NR1H2NR1H3MCL1KCNH2
SCHEMBL31439803 0.89 MCL1 (0.45) MCL1KCNH2HRH3USP30BCL2
SCHEMBL29523919 0.88 NR1H2 (0.47) P2RX3NR1H2NR1H3MCL1KCNH2
SCHEMBL30530834 0.88 NR1H2 (0.47) P2RX3NR1H2NR1H3MCL1KCNH2
SCHEMBL24739408 0.88 HRH3 (0.54) P2RX3NR1H2NR1H3MCL1KCNH2
SCHEMBL13481692 0.88 P2RX3 (0.51) P2RX3NR1H2NR1H3MCL1KCNH2
SCHEMBL12589826 0.88 P2RX3 (0.51) P2RX3NR1H2NR1H3MCL1KCNH2
SCHEMBL1198567 0.88 P2RX3 (0.51) P2RX3NR1H2NR1H3MCL1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023237457-A1 INDAZOLE MACROCYCLES FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. HOFFMANN-LA ROCHE AG (CH) 2023-12-14 WO disclosed