SCHEMBL2694565

SCHEMBL2694565

CC(C)CN1CCC2(CC1)CN(C(=O)c1ccc(CN(Cc3nccn3C)Cc3nccn3C)cc1)CCO2

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 15/20 0.45
CHRM3 P20309 15/20 0.45
CYP2D6 P10635 4/20 0.42
CYP3A4 P08684 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.38
CBLB Q13191 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14856686 0.93 CHRM2 (0.43) CHRM2CHRM3CBLB
SCHEMBL2696738 0.93 CXCR4 (0.47) CHRM2CHRM3CYP2D6CYP3A4ALDH1A1
SCHEMBL2695080 0.89 CHRM2 (0.45) CHRM2CHRM3CBLB
SCHEMBL2695556 0.87 CYP2D6 (0.53) CYP2D6CYP3A4ALDH1A1MAPK1
SCHEMBL2694068 0.87 CHRM2 (0.41) CHRM2CHRM3CBLB
SCHEMBL2695355 0.85 CYP2D6 (0.60) CYP2D6CYP3A4ALDH1A1MAPK1
SCHEMBL2695611 0.84 CXCR4 (0.53) CHRM2CHRM3CYP2D6CYP3A4ALDH1A1
SCHEMBL2692570 0.82 CXCR4 (0.44) CHRM2CHRM3CBLB
SCHEMBL2692731 0.81 CXCR4 (0.47) CHRM2CHRM3CBLB
SCHEMBL2692456 0.80 CXCR4 (0.55) CYP2D6CYP3A4ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8519124-B2 Chemokine receptor antagonists and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2013-08-27 US claimed
EP-1961744-B1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO (JP) 2013-04-17 EP claimed
US-8519124-B2 Chemokine receptor antagonists and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2013-08-27 US disclosed
EP-1961744-B1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO (JP) 2013-04-17 EP disclosed
US-20120207765-A1 CHEMOKINE RECEPTOR ANTAGONISTS AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2012-08-16 US disclosed
US-8168783-B2 Chemokine receptor antagonists and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2012-05-01 US disclosed
US-20090169567-A1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD., (JP) 2009-07-02 US disclosed
EP-1961744-A1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2008-08-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090169567-A1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF CXCR4, CXCL12, CXCR3 CHRM2 759/4885CHRM3 767/4885CYP2D6 2687/4885
US-20120207765-A1 CHEMOKINE RECEPTOR ANTAGONISTS AND USE THEREOF CXCR4, CXCR3, CXCR1 CHRM2 798/4885CHRM3 736/4885CYP2D6 2851/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.