SCHEMBL2695352

SCHEMBL2695352

CC(C)CN1CCC2(CCCN(Cc3ccc(C(=O)N(Cc4ncc[nH]4)Cc4ncc[nH]4)cc3)C2)CC1

nearest known ligand 0.87

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 3/20 0.87
OPRD1 P41143 1/20 0.47
CYP3A4 P08684 14/20 0.46
CYP2D6 P10635 9/20 0.46
CYP1A2 P05177 4/20 0.46
CYP2C9 P11712 7/20 0.43
CYP2C19 P33261 3/20 0.43
KDM1A O60341 1/20 0.43
MAOB P27338 1/20 0.43
RCOR1 Q9UKL0 1/20 0.43
USP2 O75604 2/20 0.42
ALDH1A1 P00352 5/20 0.42
TSHR P16473 2/20 0.42
CASP1 P29466 1/20 0.41
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2693586 0.97 CXCR4 (0.93) CXCR4OPRD1CYP3A4CYP2D6CYP1A2
SCHEMBL1793937 0.97 CXCR4 (0.93) CXCR4OPRD1CYP3A4CYP2D6CYP1A2
SCHEMBL2694483 0.93 CXCR4 (1.00) CXCR4OPRD1CYP3A4CYP2D6CYP1A2
SCHEMBL2695642 0.93 CXCR4 (0.90) CXCR4OPRD1CYP3A4CYP2D6CYP1A2
SCHEMBL2695823 0.91 CXCR4 (0.93) CXCR4OPRD1CYP3A4CYP2D6CYP1A2
SCHEMBL2697475 0.91 CXCR4 (0.90) CXCR4OPRD1CYP3A4CYP2D6CYP2C9
SCHEMBL2694625 0.90 CXCR4 (0.80) CXCR4OPRD1CYP3A4CYP2D6CYP1A2
SCHEMBL1793461 0.89 CXCR4 (0.71) CXCR4OPRD1CYP3A4CYP2D6CYP1A2
SCHEMBL2695486 0.89 CXCR4 (0.79) CXCR4OPRD1CYP3A4CYP2D6CYP1A2
SCHEMBL1798887 0.89 CXCR4 (0.73) CXCR4OPRD1CYP3A4CYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8519124-B2 Chemokine receptor antagonists and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2013-08-27 US claimed
EP-1961744-B1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO (JP) 2013-04-17 EP claimed
US-8519124-B2 Chemokine receptor antagonists and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2013-08-27 US disclosed
EP-1961744-B1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO (JP) 2013-04-17 EP disclosed
US-20120207765-A1 CHEMOKINE RECEPTOR ANTAGONISTS AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2012-08-16 US disclosed
US-8168783-B2 Chemokine receptor antagonists and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2012-05-01 US disclosed
US-20090169567-A1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD., (JP) 2009-07-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090169567-A1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF CXCR4, CXCL12, CXCR3 CXCR4 1/4885OPRD1 2003/4885CYP3A4 3747/4885
US-20120207765-A1 CHEMOKINE RECEPTOR ANTAGONISTS AND USE THEREOF CXCR4, CXCR3, CXCR1 CXCR4 1/4885OPRD1 1440/4885CYP3A4 4052/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.