SCHEMBL2695409

SCHEMBL2695409

CC(C)CN1CCC2(CC1)CN(C(=O)c1ccc(CN(Cc3ncc[nH]3)Cc3ncc[nH]3)cc1)C2

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 2/20 0.62
CYP2D6 P10635 12/20 0.51
CYP3A4 P08684 9/20 0.51
ALDH1A1 P00352 2/20 0.51
CYP1A2 P05177 4/20 0.46
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
USP2 O75604 3/20 0.46
HIF1A Q16665 1/20 0.46
HSD17B10 Q99714 1/20 0.40
CYP2C19 P33261 1/20 0.40
HRH3 Q9Y5N1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2691751 0.95 CXCR4 (0.63) CXCR4CYP2D6CYP3A4ALDH1A1CYP1A2
SCHEMBL2695977 0.94 CXCR4 (0.60) CXCR4CYP2D6CYP3A4ALDH1A1CYP1A2
SCHEMBL2692849 0.93 CXCR4 (0.61) CXCR4CYP2D6CYP3A4ALDH1A1CYP1A2
SCHEMBL2693802 0.93 CXCR4 (0.62) CXCR4CYP2D6CYP3A4ALDH1A1CYP1A2
SCHEMBL2696569 0.89 CXCR4 (0.56) CXCR4CYP2D6CYP3A4ALDH1A1CYP1A2
SCHEMBL2692456 0.88 CXCR4 (0.55) CXCR4CYP2D6CYP3A4ALDH1A1CYP1A2
SCHEMBL2694823 0.87 CXCR4 (0.49) CXCR4CYP2D6CYP3A4ALDH1A1CYP1A2
SCHEMBL2697323 0.87 CXCR4 (0.53) CXCR4CYP2D6CYP3A4ALDH1A1CYP1A2
SCHEMBL2694235 0.86 CXCR4 (0.59) CXCR4CYP2D6CYP3A4ALDH1A1CYP1A2
SCHEMBL2695611 0.86 CXCR4 (0.53) CXCR4CYP2D6CYP3A4ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8519124-B2 Chemokine receptor antagonists and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2013-08-27 US claimed
EP-1961744-B1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO (JP) 2013-04-17 EP claimed
US-8519124-B2 Chemokine receptor antagonists and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2013-08-27 US disclosed
US-8519124-B2 Chemokine receptor antagonists and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2013-08-27 US disclosed
EP-1961744-B1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO (JP) 2013-04-17 EP disclosed
US-20120207765-A1 CHEMOKINE RECEPTOR ANTAGONISTS AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2012-08-16 US disclosed
US-20120207765-A1 CHEMOKINE RECEPTOR ANTAGONISTS AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2012-08-16 US disclosed
US-8168783-B2 Chemokine receptor antagonists and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2012-05-01 US disclosed
US-8168783-B2 Chemokine receptor antagonists and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2012-05-01 US disclosed
US-8168783-B2 Chemokine receptor antagonists and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2012-05-01 US disclosed
US-20090169567-A1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD., (JP) 2009-07-02 US disclosed
US-20090169567-A1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD., (JP) 2009-07-02 US disclosed
US-20090169567-A1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD., (JP) 2009-07-02 US disclosed
EP-1961744-A1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2008-08-27 EP disclosed
EP-1961744-A1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2008-08-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090169567-A1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF CXCR4, CXCL12, CXCR3 CXCR4 1/4885CYP2D6 2687/4885CYP3A4 3747/4885
US-20120207765-A1 CHEMOKINE RECEPTOR ANTAGONISTS AND USE THEREOF CXCR4, CXCR3, CXCR1 CXCR4 1/4885CYP2D6 2851/4885CYP3A4 4052/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.