Ciprofloxacin

Ciprofloxacin

SCHEMBL27004

Cl.O.O=C(O)c1cn(C2CC2)c2cc(N3CCNCC3)c(F)cc2c1=O

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

gyrAgyrBparCparE

The experimentally established mechanism targets of Ciprofloxacin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.96
ALDH1A1 P00352 6/20 0.96
LMNA P02545 5/20 0.96
HPGD P15428 4/20 0.96
HSD17B10 Q99714 4/20 0.96
CYP1A2 P05177 1/20 0.96
TOP2A P11388 1/20 0.96
CYP2C9 P11712 1/20 0.96
TOP2B Q02880 1/20 0.96
MAPT P10636 1/20 0.70
HTT P42858 2/20 0.65
BRD4 O60885 1/20 0.65
TSHR P16473 1/20 0.65
CYP2J2 P51589 1/20 0.65
NPSR1 Q6W5P4 1/20 0.65
PIK3CG P48736 7/20 0.61
PIK3CD O00329 5/20 0.61
PIK3R1 P27986 5/20 0.61
PIK3CA P42336 5/20 0.61
SMN1; SMN2 Q16637 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ciprofloxacin SCHEMBL1281819 1.00 KDM4E (0.96) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL2325952 1.00 KDM4E (0.96) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL184706 1.00 KDM4E (0.96) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL8530004 1.00 KDM4E (0.96) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL2636760 1.00 KDM4E (0.96) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL23064249 1.00 KDM4E (0.96) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL2465661 0.99 KDM4E (0.98) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL42310 0.99 KDM4E (0.98) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL7994990 0.99 KDM4E (0.98) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL9788110 0.99 KDM4E (0.98) KDM4EALDH1A1LMNAHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 12953 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122079427-A Method for degrading organic pollutants by coupling nano-confinement catalytic membrane with micro-nano bubbles 2026-05-26 CN claimed
WO-2026090462-A1 STABLE CIPROFLOXACIN COMPOSITIONS HIKMA PHARMACEUTICALS USA INC. (US) 2026-04-30 WO claimed
EP-4724839-A2 CONTACT LENSES INCLUDING MEDICAMENTS AND METHODS OF MAKING AND USING SAME INCLUDING SLOW RELEASE OF GLAUCOMA TREATING DRUGS AND COMFORT ENHANCING DRUGS Mediprint Ophthalmics Inc. (US) 2026-04-15 EP claimed
US-20260090984-A1 CONTACT LENSES INCLUDING MEDICAMENTS AND METHODS OF MAKING AND USING SAME INCLUDING SLOW RELEASE OF GLAUCOMA TREATING DRUGS AND COMFORT ENHANCING DRUGS MEDIPRINT OPHTHALMICS INC. (US) 2026-04-02 US claimed
US-20260076872-A1 POLYMER VIALS WITH SUBSTANTIALLY FLAT BOTTOMS AND INJECTION STRETCH BLOW MOLDING METHODS FOR MAKING THE SAME SIO2 MEDICAL PRODUCTS LLC (US) 2026-03-19 US claimed
US-20260027140-A1 COMPOSITIONS AND METHODS FOR TREATING AND AMELIORATING RESPIRATORY CONDITIONS AND INFLAMMATION OF MUCOSA ATOPIC MEDICAL INC (US) 2026-01-29 US claimed
US-12452700-B2 Setting system and setting method for setting base station device RAKUTEN SYMPHONY, INC. (JP) 2025-10-21 US claimed
US-20250242092-A1 SiOx BARRIER FOR PHARMACEUTICAL PACKAGE AND COATING PROCESS SIO2 MEDICAL PRODUCTS INC (US) 2025-07-31 US claimed
US-20250244340-A1 DIAGNOSING AND TREATING A PATHOLOGICAL CONDITION OF THE INTESTINAL TRACT MAGNOSTICS LIMITED (IE) 2025-07-31 US claimed
CN-120115168-A Aluminum-based nano-oxidase and preparation method and application thereof 广东工业大学 2025-06-10 CN claimed
US-5700410-A Method of manufacturing wax matrices NIPPON SHINYAKU CO., LTD. (JP) 1997-12-23 US claimed
EP-0580860-B1 METHOD OF MANUFACTURING SOLID DISPERSION NIPPON SHINYAKU CO LTD (JP) 1997-10-22 EP claimed
WO-1997005880-A1 AQUEOUS COMPOSITIONS CONTAINING CIPROFLOXACINE, AND RELATED USE AND PROCESS BAYVIT, S.A. (ES) 1997-02-20 WO claimed
EP-0696201-A4 SUPPLEMENTED AND UNSUPPLEMENTED TISSUE SEALANTS, METHODS OF THEIR PRODUCTION AND USE AMERICAN NAT RED CROSS (US) 1996-06-26 EP claimed
EP-0696201-A1 SUPPLEMENTED AND UNSUPPLEMENTED TISSUE SEALANTS, METHODS OF THEIR PRODUCTION AND USE AMERICAN NATIONAL RED CROSS (US) 1996-02-14 EP claimed
CN-1115641-A Prepn of cyclopropyloxacini injecta NORTHEAST GENERAL PHARMACEUTIC (CN) 1996-01-31 CN claimed
WO-1994020133-A1 SUPPLEMENTED AND UNSUPPLEMENTED TISSUE SEALANTS, METHODS OF THEIR PRODUCTION AND USE THE AMERICAN NATIONAL RED CROSS (US) 1994-09-15 WO claimed
US-5286754-A Microcrystalline cellulose, moist starch, crosslinked polyvinylpyrrolidone, silicon dixode and magnesium stearate BAYER AKTIENGESELLSCHAFT (DE) 1994-02-15 US claimed
EP-0230881-B1 PHARMACEUTICAL PREPARATIONS CONTAINING CIPROFLOXACIN BAYER AG (DE) 1991-05-15 EP claimed
EP-0394553-A2 Use of fluorine containing pyridone carboxylic acid derivatives for preparing a medicament for the treatment of HIV infections DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1990-10-31 EP claimed