Ciprofloxacin

Ciprofloxacin

SCHEMBL8530004

Cl.Cl.O.O.O=C(O)c1cn(C2CC2)c2cc(N3CCNCC3)c(F)cc2c1=O.O=C(O)c1cn(C2CC2)c2cc(N3CCNCC3)c(F)cc2c1=O

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

gyrAgyrBparCparE

The experimentally established mechanism targets of Ciprofloxacin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.96
ALDH1A1 P00352 6/20 0.96
LMNA P02545 5/20 0.96
HPGD P15428 4/20 0.96
HSD17B10 Q99714 4/20 0.96
CYP1A2 P05177 1/20 0.96
TOP2A P11388 1/20 0.96
CYP2C9 P11712 1/20 0.96
TOP2B Q02880 1/20 0.96
MAPT P10636 1/20 0.70
HTT P42858 2/20 0.65
BRD4 O60885 1/20 0.65
TSHR P16473 1/20 0.65
CYP2J2 P51589 1/20 0.65
NPSR1 Q6W5P4 1/20 0.65
PIK3CG P48736 7/20 0.61
PIK3CD O00329 5/20 0.61
PIK3R1 P27986 5/20 0.61
PIK3CA P42336 5/20 0.61
SMN1; SMN2 Q16637 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ciprofloxacin SCHEMBL1281819 1.00 KDM4E (0.96) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL2325952 1.00 KDM4E (0.96) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL184706 1.00 KDM4E (0.96) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL27004 1.00 KDM4E (0.96) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL2636760 1.00 KDM4E (0.96) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL23064249 1.00 KDM4E (0.96) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL2465661 0.99 KDM4E (0.98) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL42310 0.99 KDM4E (0.98) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL7994990 0.99 KDM4E (0.98) KDM4EALDH1A1LMNAHPGDHSD17B10
Ciprofloxacin SCHEMBL9788110 0.99 KDM4E (0.98) KDM4EALDH1A1LMNAHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190204229-A1 Low Energy Laser Spectroscopy LELS HUDSON GUSTAV (US) 2019-07-04 US disclosed
US-10324037-B2 Low energy laser spectroscopy LELS HUDSON GUSTAV (US) 2019-06-18 US disclosed
US-20160290922-A1 Low Energy Laser Spectroscopy HUDSON GUSTAV (US) 2016-10-06 US disclosed
US-20160161411-A1 Low Energy Laser Spectroscopy LELS HUDSON GUSTAV (US) 2016-06-09 US disclosed
WO-2012110971-A2 METHOD AND COMPOSITION TO RETARD SORPTION OF PRESERVATIVES TO PLASTICS PROMED EXPORTS PVT. LTD. (IN) 2012-08-23 WO disclosed
US-5814335-A FORMING LIPOSOME FROM MIXTURE OF SPHINGOMYELIN AND CHOLESTEROL IN BUFFERED AQUEOUS SOLUTION, SUSPENDING IN SECOND SOLUTION INEX PHARMACEUTICALS CORPORATION (CA) 1998-09-29 US disclosed
US-5741516-A LIPOSOMAL FORMULATIONS HAVING EXTENDED CIRCULATION TIME IN VIVO AND INCREASED DRUG RETENTION COMPRISED OF SPHINGOMYELIN AND CHOLESTEROL; ACIDIC INTRALIPOSOMAL PH INEX PHARMACEUTICALS CORPORATION (CA) 1998-04-21 US disclosed