SCHEMBL2716657

SCHEMBL2716657

CCc1nc(N)cc(C(C)C)n1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 9/20 0.52
NOS3 P29474 7/20 0.52
NOS1 P29475 6/20 0.52
MAPT P10636 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
HRH3 Q9Y5N1 5/20 0.35
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
HTR1B P28222 1/20 0.30
HTR2B P41595 1/20 0.30
GPR65 Q8IYL9 1/20 0.30
HRH4 Q9H3N8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28267332 0.80 MAPT (0.56) NOS2NOS3NOS1MAPTTDP1
SCHEMBL17995540 0.78 ESR1 (0.36) NOS2NOS3NOS1
SCHEMBL12015758 0.74 NOS2 (0.59) NOS2NOS3NOS1HRH3MEN1
SCHEMBL798760 0.73 PDE2A (0.33) NOS2NOS3NOS1ALDH1A1
SCHEMBL26816606 0.73 NOS2 (0.41) NOS2NOS3NOS1MAPTTDP1
SCHEMBL7769935 0.72 NOS2 (0.63) NOS2NOS3NOS1HRH3MEN1
SCHEMBL18011660 0.72 NOS2 (0.48) NOS2NOS3NOS1MAPTTDP1
SCHEMBL2719526 0.72 NOS2 (0.57) NOS2NOS3NOS1MAPTTDP1
SCHEMBL2717960 0.72 NOS2 (0.57) NOS2NOS3NOS1HRH3MEN1
SCHEMBL21937782 0.72 CYP3A4 (0.57) NOS2NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012061337-A1 FGFR2 MODULATORS EXELIXIS, INC. (US) 2012-05-10 WO disclosed