SCHEMBL27190835

SCHEMBL27190835

CN(C)C=C(C(=O)O)C(=O)CC(=O)O

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.33
SRR Q9GZT4 1/20 0.33
KDM4E B2RXH2 1/20 0.32
TSHR P16473 1/20 0.32
ALOX15 P16050 1/20 0.30
HSD17B10 Q99714 1/20 0.30
KDM7A Q6ZMT4 1/20 0.30
PHF8 Q9UPP1 1/20 0.30
KDM2A Q9Y2K7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26914828 1.00 LDHA (0.33) LDHASRRKDM4ETSHRALOX15
SCHEMBL29191376 0.82 EGLN1 (0.35) KDM4E
SCHEMBL29191375 0.82 MGAM (0.37) TSHRHSD17B10
SCHEMBL21355685 0.81 EGLN1 (0.46) KDM4EKDM7APHF8KDM2A
SCHEMBL3355710 0.80 FFAR3 (0.33)
SCHEMBL3355714 0.80 FFAR3 (0.33)
SCHEMBL17610271 0.80 FFAR3 (0.33)
SCHEMBL25242898 0.78 TSHR (0.32) TSHR
SCHEMBL28995635 0.78 TSHR (0.32) TSHR
SCHEMBL22531952 0.78 ABAT (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4346815-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE Schrödinger, Inc. (US) 2024-04-10 EP disclosed
CN-117715642-A Heterocyclic compounds and methods of use 薛定谔公司 2024-03-15 CN disclosed
CN-117357650-A Pharmaceutical composition comprising SOS1 inhibitor 武汉人福创新药物研发中心有限公司 2024-01-09 CN disclosed
WO-2022251497-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE SCHRÖDINGER, INC. (US) 2022-12-01 WO disclosed