SCHEMBL2719956

SCHEMBL2719956

CS(=O)(=O)Cc1c(-c2ccccc2)c(CCNc2ncnc(N)c2C#N)nc2ccc(F)cc12

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 20/20 0.58
PIK3CG P48736 20/20 0.58
PIK3CB P42338 19/20 0.58
PIK3CA P42336 16/20 0.58
CYP3A4 P08684 4/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2717267 0.89 PIK3CD (0.68) PIK3CDPIK3CGPIK3CBPIK3CACYP3A4
SCHEMBL2717125 0.88 PIK3CD (0.57) PIK3CDPIK3CGPIK3CBPIK3CACYP3A4
SCHEMBL2719384 0.88 PIK3CD (0.64) PIK3CDPIK3CGPIK3CBPIK3CACYP3A4
SCHEMBL2719807 0.87 PIK3CD (0.73) PIK3CDPIK3CGPIK3CBPIK3CACYP3A4
SCHEMBL2717151 0.86 PIK3CD (0.57) PIK3CDPIK3CGPIK3CBPIK3CACYP3A4
SCHEMBL2718353 0.84 PIK3CD (0.67) PIK3CDPIK3CGPIK3CBPIK3CACYP3A4
SCHEMBL2718432 0.84 PIK3CD (0.59) PIK3CDPIK3CGPIK3CBPIK3CACYP3A4
SCHEMBL2717745 0.83 PIK3CD (0.58) PIK3CDPIK3CGPIK3CBPIK3CACYP3A4
SCHEMBL2717233 0.83 PIK3CD (0.70) PIK3CDPIK3CGPIK3CBPIK3CACYP3A4
SCHEMBL2720033 0.83 PIK3CD (0.59) PIK3CDPIK3CGPIK3CBPIK3CACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2445900-A2 POLYCYCLIC DERIVATIVES OF PYRIDINE AND THEIR USE IN THE TREATMENT OF (INTER ALIA) RHEUMATOID ARTHRITIS AND SIMILAR DISEASES Amgen, Inc (US) 2012-05-02 EP disclosed
WO-2010151740-A2 HETEROCYCLIC COMPOUNDS AND THEIR USES AMGEN INC. (US) 2010-12-29 WO disclosed