SCHEMBL2722552

SCHEMBL2722552

COc1cc2nc(CF)[nH]c(=O)c2cc1OC

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.67
GAA P10253 1/20 0.67
TDP1 Q9NUW8 1/20 0.60
LMNA P02545 4/20 0.57
MAPK1 P28482 2/20 0.57
USP2 O75604 1/20 0.57
ALDH1A1 P00352 1/20 0.57
ALOX15 P16050 1/20 0.57
MAPT P10636 2/20 0.56
PDE3B Q13370 3/20 0.51
PDE3A Q14432 3/20 0.51
TUBB4A P04350 1/20 0.50
TUBB P07437 1/20 0.50
TUBA3C P0DPH7 1/20 0.50
TUBA1B P68363 1/20 0.50
TUBA4A P68366 1/20 0.50
TUBB4B P68371 1/20 0.50
TUBB3 Q13509 1/20 0.50
TUBB2A Q13885 1/20 0.50
TUBB8 Q3ZCM7 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25112482 0.89 KDM4E (0.54) KDM4EGAATDP1LMNAMAPK1
SCHEMBL27167377 0.86 KDM4E (0.72) KDM4EGAATDP1LMNAMAPK1
SCHEMBL2722306 0.85 KDM4E (0.67) KDM4EGAATDP1LMNAMAPK1
SCHEMBL24792433 0.85 KDM4E (0.67) KDM4EGAATDP1LMNAMAPK1
SCHEMBL29900596 0.85 KDM4E (0.67) KDM4EGAATDP1LMNAMAPK1
SCHEMBL6120242 0.82 KDM4E (0.71) KDM4EGAATDP1LMNAMAPK1
SCHEMBL28875071 0.80 KDM4E (0.64) KDM4EGAATDP1LMNAMAPK1
SCHEMBL6128121 0.78 KDM4E (0.62) KDM4EGAATDP1LMNAMAPK1
SCHEMBL23882078 0.77 KDM4E (0.54) KDM4EGAATDP1LMNAMAPK1
SCHEMBL31716637 0.77 KDM4E (0.57) KDM4EGAATDP1LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012052556-A1 NOVEL HALOALKOXYQUINAZOLINES, AND PREPARATION AND USE THEREOF UNIVERSITÄT LEIPZIG (DE) 2012-04-26 WO disclosed
WO-2012052556-A1 NOVEL HALOALKOXYQUINAZOLINES, AND PREPARATION AND USE THEREOF UNIVERSITÄT LEIPZIG (DE) 2012-04-26 WO disclosed