SCHEMBL28875071

SCHEMBL28875071

CCCCCc1nc2cc(OC)c(OC)cc2c(=O)[nH]1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.64
GAA P10253 1/20 0.64
MAPK1 P28482 2/20 0.56
USP2 O75604 1/20 0.56
ALDH1A1 P00352 1/20 0.56
ALOX15 P16050 1/20 0.56
TDP1 Q9NUW8 1/20 0.55
PARP1 P09874 1/20 0.53
LMNA P02545 4/20 0.53
MAPT P10636 2/20 0.52
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
THRB P10828 1/20 0.47
CASP1 P29466 1/20 0.47
HBB P68871 1/20 0.47
TUBB4A P04350 1/20 0.46
TUBB P07437 1/20 0.46
TUBA3C P0DPH7 1/20 0.46
TUBA1B P68363 1/20 0.46
TUBA4A P68366 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27167377 0.84 KDM4E (0.72) KDM4EGAAMAPK1USP2ALDH1A1
SCHEMBL2722552 0.80 KDM4E (0.67) KDM4EGAAMAPK1USP2ALDH1A1
SCHEMBL2722306 0.80 KDM4E (0.67) KDM4EGAAMAPK1USP2ALDH1A1
SCHEMBL24792433 0.80 KDM4E (0.67) KDM4EGAAMAPK1USP2ALDH1A1
SCHEMBL29900596 0.80 KDM4E (0.67) KDM4EGAAMAPK1USP2ALDH1A1
SCHEMBL6120242 0.78 KDM4E (0.71) KDM4EGAAMAPK1USP2ALDH1A1
SCHEMBL28307055 0.78 PARP1 (0.41) KDM4EGAAMAPK1PARP1
SCHEMBL7415916 0.77 PARP1 (0.63) KDM4EGAAUSP2PARP1LMNA
SCHEMBL19846637 0.76 PARP1 (0.60) PARP1
SCHEMBL2266470 0.76 PDE10A (0.55) KDM4EGAAALDH1A1TDP1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110041306-A 4- hydroxyl -2- quinolone-nitrogen-(4- quinazolinone) -3- carboxamides derivatives 中国医学科学院药物研究所 2019-07-23 CN disclosed