SCHEMBL27228

SCHEMBL27228

c1ccc(CCNCc2ccccc2)cc1

nearest known ligand 0.95

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.95
MAPT P10636 1/20 0.95
MEN1 O00255 1/20 0.76
KMT2A Q03164 1/20 0.76
TDP1 Q9NUW8 1/20 0.76
SIGMAR1 Q99720 7/20 0.72
BCHE P06276 1/20 0.67
MAOA P21397 1/20 0.67
KDM4E B2RXH2 1/20 0.65
ALDH1A1 P00352 1/20 0.65
CA12 O43570 1/20 0.65
CA1 P00915 1/20 0.65
CA2 P00918 1/20 0.65
CA4 P22748 1/20 0.65
CA9 Q16790 1/20 0.65
CHRM2 P08172 1/20 0.64
MPO P05164 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25432637 0.98 GAA (0.91) GAAMAPTMEN1KMT2ATDP1
Hydrochloric Acid SCHEMBL1983401 0.98 GAA (1.00) GAAMAPTMEN1KMT2ATDP1
SCHEMBL11881258 0.98 GAA (0.91) GAAMAPTMEN1KMT2ATDP1
Ammonia Solution, Strong SCHEMBL23581968 0.98 GAA (0.91) GAAMAPTMEN1KMT2ATDP1
SCHEMBL3272134 0.98 GAA (0.91) GAAMAPTMEN1KMT2ATDP1
Ethylenediamine SCHEMBL9304893 0.91 GAA (0.80) GAAMAPTMEN1KMT2ATDP1
Bicarbonate SCHEMBL11575509 0.91 GAA (0.80) GAAMAPTMEN1KMT2ATDP1
SCHEMBL10060315 0.91 GAA (0.80) GAAMAPTMEN1KMT2ATDP1
Diethylamine SCHEMBL7882261 0.89 GAA (0.77) GAAMAPTMEN1KMT2ATDP1
SCHEMBL10133040 0.89 GAA (0.77) GAAMAPTMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 19592 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026044024-A1 COMPOSITIONS COMPRISING COMBINATIONS OF PHARMACEUTICALLY ACCEPTABLE SALTS AND OTHER DERIVATIVES OF GLUCAGON-LIKE PEPTIDE-1 RECEPTOR AGONIST AND PHARMACEUTICALLY ACCEPTABLE SALTS AND OTHER DERIVATIVES OF AMYLIN ANALOG, AND USES THEREOF I2O THERAPEUTICS, INC. (US) 2026-02-26 WO claimed
EP-3807293-B1 PEPTIDES HAVING INHIBITORY ACTIVITY ON NEURONAL EXOCYTOSIS ACRAF (IT) 2026-01-14 EP claimed
EP-3807294-B1 PEPTIDES HAVING INHIBITORY ACTIVITY ON MUSCARINIC RECEPTOR M3 ACRAF (IT) 2026-01-14 EP claimed
US-20250387385-A1 TREATMENT FOR GLOMERULAR DISEASES ZYDUS LIFESCIENCES LIMITED (IN) 2025-12-25 US claimed
EP-4660194-A1 SALT AND CRYSTAL FORM OF CYCLOALKENE COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF Jiangsu Hansoh Pharmaceutical Group Co., Ltd. (CN) 2025-12-10 EP claimed
US-20250353840-A1 SOLID FORMS OF (Z)-4-(5-((3-BENZYL-4-OXO-2-THIOXOTHIAZOLIDIN-5-YLIDENE) METHYL)FURAN-2-YL)BENZOIC ACID ATEGRIN INC (US) 2025-11-20 US claimed
US-12421264-B2 Compounds and methods for the treatment of pathogenic Neisseria INSTITUT NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CA) 2025-09-23 US claimed
US-12390402-B2 High-content and sustained-release retinoid capsule, and composition for reducing wrinkles, containing same LG HOUSEHOLD & HEALTHCARE LTD. (KR) 2025-08-19 US claimed
US-12377035-B2 Peptides for inhibiting cholinergic calcitonin gene-related peptide (CGRP) and acetylcholine (ACH) release or inhibiting sensitization-mediated by TRPV1-mediated excitability in sensory neurons and methods of use thereof AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO—A.C.R.A.F. S.p.A. (IT) 2025-08-05 US claimed
EP-4565233-A1 TREATMENT FOR APLASTIC ANEMIA (AA) Zydus Lifesciences Limited (IN) 2025-06-11 EP claimed
US-4029806-A Nitro-β-lactam antibiotics and processes for their preparation and use BAYER AKTIENGESELLSCHAFT (DT) 1977-06-14 US claimed
US-4012518-A PENICILLIN DERIVATIVES AS GROWTH AND FEED UTILIZATION PROMOTERS IN ANIMALS BAYER AKTIENGESELLSCHAFT (DT) 1977-03-15 US claimed
US-4001218-A BACTERICIDES BAYER AKTIENGESELLSCHAFT (DT) 1977-01-04 US claimed
US-3993642-A Penicillins BAYER AKTIENGESELLSCHAFT (DT) 1976-11-23 US claimed
US-3993770-A Penicillins BAYER AKTIENGESELLSCHAFT (DT) 1976-11-23 US claimed
US-3988327-A 7-(α-SULFOACYLAMIDO)CEPHALOSPORANIC ACIDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JA) 1976-10-26 US claimed
US-3982011-A ANTIBIOTICS, ANIMAL GROWTH PROMOTERS BAYER AKTIENGESELLSCHAFT (DT) 1976-09-21 US claimed
US-3974288-A ANTIBACTERIAL ACTIVITY BAYER AKTIENGESELLSCHAFT (DT) 1976-08-10 US claimed
US-3944544-A BACTERICIDE E. R. SQUIBB & SONS, INC. (US) 1976-03-16 US claimed
US-3931153-A BACTERICIDE BAYER AKTIENGESELLSCHAFT (DT) 1976-01-06 US claimed