SCHEMBL2723536

SCHEMBL2723536

FC(F)(F)O/C=C/c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.44
NFE2L2 Q16236 4/20 0.43
CYP1A1 P04798 1/20 0.41
CYP1B1 Q16678 1/20 0.41
TRPA1 O75762 2/20 0.39
ALDH1A1 P00352 2/20 0.38
LMNA P02545 2/20 0.38
CYP19A1 P11511 1/20 0.38
MAOA P21397 1/20 0.38
ALOX5 P09917 1/20 0.38
MAPK1 P28482 1/20 0.38
IDO1 P14902 2/20 0.38
HDAC3 O15379 1/20 0.37
TNKS O95271 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HCAR2 Q8TDS4 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2723539 1.00 MAOB (0.44) MAOBNFE2L2CYP1A1CYP1B1TRPA1
SCHEMBL29905579 0.79 MAOB (0.38) MAOBNFE2L2CYP1A1CYP1B1TRPA1
SCHEMBL7770617 0.77 MAOB (0.44) MAOBNFE2L2CYP1A1CYP1B1TRPA1
SCHEMBL187273 0.77 MAOB (0.44) MAOBNFE2L2CYP1A1CYP1B1TRPA1
SCHEMBL8092474 0.77 MAOB (0.35) MAOBNFE2L2CYP1A1CYP1B1TRPA1
SCHEMBL821619 0.76 ALDH1A1 (0.36) MAOBNFE2L2CYP1A1CYP1B1TRPA1
SCHEMBL8996775 0.76 MAOB (0.42) MAOBNFE2L2TRPA1ALDH1A1LMNA
SCHEMBL15709852 0.73 MAOB (0.50) MAOBNFE2L2TRPA1ALDH1A1LMNA
SCHEMBL29716694 0.72 MAOB (0.39) MAOBNFE2L2CYP1A1CYP1B1TRPA1
SCHEMBL28560204 0.72 MAPK1 (0.50) MAOBNFE2L2TRPA1ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054782-A2 FLUOROALKOXYLATION OF ORGANIC COMPOUNDS PRESIDENTS AND FELLOWS OF HARVARD COLLEGE (US) 2012-04-26 WO claimed
WO-2012054782-A2 FLUOROALKOXYLATION OF ORGANIC COMPOUNDS PRESIDENTS AND FELLOWS OF HARVARD COLLEGE (US) 2012-04-26 WO disclosed