SCHEMBL2723947

SCHEMBL2723947

COc1ccc(-c2onc(-c3ccccc3Cl)c2-c2ccccc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.59
PTGS1 P23219 1/20 0.59
HSP90AA1 P07900 3/20 0.48
GPBAR1 Q8TDU6 1/20 0.47
LMNA P02545 2/20 0.46
MAPT P10636 1/20 0.46
THRB P10828 1/20 0.44
S1PR1 P21453 1/20 0.44
NR1H4 Q96RI1 1/20 0.44
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
GAA P10253 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9956787 0.91 HSP90AA1 (0.51) PTGS2PTGS1HSP90AA1GPBAR1LMNA
SCHEMBL2722592 0.88 PTGS1 (0.69) PTGS2PTGS1GPBAR1LMNAMAPT
SCHEMBL4549984 0.88 PTGS2 (0.50) PTGS2PTGS1HSP90AA1GPBAR1LMNA
SCHEMBL2723070 0.87 TP53 (0.47) PTGS2PTGS1HSP90AA1GPBAR1LMNA
SCHEMBL2720986 0.83 PTGS1 (0.52) PTGS2PTGS1HSP90AA1GPBAR1LMNA
SCHEMBL2721067 0.83 GPBAR1 (0.47) PTGS2PTGS1HSP90AA1GPBAR1LMNA
SCHEMBL2732395 0.83 PTGS1 (0.59) PTGS2PTGS1LMNAMAPTS1PR1
SCHEMBL2721647 0.83 PTGS2 (0.45) PTGS2PTGS1HSP90AA1GPBAR1LMNA
SCHEMBL5729672 0.79 PTGS2 (0.70) PTGS2PTGS1
SCHEMBL10080406 0.79 PTGS1 (0.65) PTGS2PTGS1GPBAR1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012052395-A1 ISOXAZOLE DERIVATIVES USED AS OESTROGEN MODULATORS N. V. ORGANON (NL) 2012-04-26 WO disclosed