SCHEMBL2725908

SCHEMBL2725908

Cc1coc(-c2cc(-c3ncco3)cc(C(N)=O)c2C)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 2/20 0.39
PIK3CB P42338 1/20 0.36
GLRA3 O75311 1/20 0.36
GLRB P48167 1/20 0.36
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
IRAK4 Q9NWZ3 5/20 0.34
IL2 P60568 1/20 0.34
CFTR P13569 1/20 0.33
BRD4 O60885 1/20 0.33
HCRTR1 O43613 2/20 0.32
HCRTR2 O43614 2/20 0.32
AOC3 Q16853 2/20 0.32
PKMYT1 Q99640 1/20 0.32
TUBB4A P04350 1/20 0.31
TUBB P07437 1/20 0.31
TUBA3C P0DPH7 1/20 0.31
TUBA1B P68363 1/20 0.31
TUBA4A P68366 1/20 0.31
TUBB4B P68371 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2725903 0.83 PIK3CB (0.36) TGFBR1PIK3CBGLRA3GLRBCCNC
SCHEMBL3347772 0.83 GLRA3 (0.44) PIK3CBGLRA3GLRBCCNCCDK8
SCHEMBL2724735 0.82 PARP1 (0.39) TGFBR1PIK3CBGLRA3GLRBCCNC
SCHEMBL2726265 0.81 TGFBR1 (0.38) TGFBR1PIK3CBGLRA3GLRBCCNC
SCHEMBL2728043 0.78 KDM4B (0.39) TGFBR1PIK3CBGLRA3GLRBIL2
SCHEMBL3353479 0.73 CFTR (0.43) PIK3CBGLRA3GLRBCCNCCDK8
SCHEMBL2725910 0.73 CFTR (0.43) PIK3CBGLRA3GLRBCCNCCDK8
SCHEMBL2724726 0.73 PARP1 (0.39) PIK3CBGLRA3GLRBIL2CFTR
SCHEMBL10320333 0.71 BRD4 (0.46) PIK3CBGLRA3GLRBIL2CFTR
SCHEMBL2726899 0.71 ADORA2A (0.36) TGFBR1PIK3CBGLRA3GLRBHCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed