SCHEMBL2726320

SCHEMBL2726320

O=C(N[C@H]1c2cc(N3CCNCC3)ccc2C[C@@H]1O)c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 15/20 0.50
CHRM2 P08172 13/20 0.50
CHRM4 P08173 11/20 0.50
CTSS P25774 2/20 0.45
MAOB P27338 1/20 0.45
NAMPT P43490 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2610209 0.90 CTSS (0.52) CHRM1CHRM2CHRM4CTSSMAOB
Hydrochloric Acid SCHEMBL2115298 0.89 CTSS (0.51) CHRM1CHRM2CHRM4CTSSMAOB
SCHEMBL2610207 0.88 CHRM1 (0.53) CHRM1CHRM2CHRM4CTSS
SCHEMBL2610210 0.88 CTSS (0.49) CHRM1CHRM2CHRM4CTSSMAOB
Hydrochloric Acid SCHEMBL2113656 0.87 CTSS (0.48) CHRM1CHRM2CHRM4CTSSMAOB
SCHEMBL2113051 0.86 CHRM1 (0.49) CHRM1CHRM2CHRM4CTSSNAMPT
SCHEMBL2710639 0.83 CHRM1 (0.45) CHRM1CHRM2CHRM4CTSSNAMPT
SCHEMBL2113182 0.83 CTSS (0.65) CHRM1CHRM2CHRM4CTSSNAMPT
SCHEMBL2115295 0.82 CTSS (0.55) CTSSMAOB
SCHEMBL2732555 0.82 CTSS (0.55) CTSSMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630141-A1 CATHEPSIN S INHIBITOR COMPOUNDS Eli Lilly and Company (US) 2013-08-28 EP disclosed
WO-2012054315-A1 CATHEPSIN S INHIBITOR COMPOUNDS ELI LILLY AND COMPANY (US) 2012-04-26 WO disclosed