SCHEMBL27280448

SCHEMBL27280448

COC(=O)c1c(F)cc(Br)cc1OC1CCCC1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 9/20 0.42
PDE4A P27815 7/20 0.42
PDE4B Q07343 7/20 0.42
PDE4C Q08493 7/20 0.42
KMT2A Q03164 2/20 0.41
SCN9A Q15858 1/20 0.40
POLB P06746 1/20 0.39
PDE5A O76074 1/20 0.38
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
MEN1 O00255 1/20 0.36
NPY1R P25929 1/20 0.36
NPY2R P49146 1/20 0.36
EPHX2 P34913 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20562535 0.97 PDE4D (0.40) PDE4DPDE4APDE4BPDE4CKMT2A
SCHEMBL16935328 0.86 KMT2A (0.40) PDE4DPDE4APDE4BPDE4CKMT2A
SCHEMBL27280475 0.85 SCN9A (0.44) PDE4DPDE4APDE4BPDE4CSCN9A
SCHEMBL31535452 0.85 KMT2A (0.44) PDE4DPDE4APDE4BPDE4CKMT2A
SCHEMBL27280537 0.80 PDE4D (0.42) PDE4DPDE4APDE4BPDE4CSCN9A
SCHEMBL12470349 0.79 NOTUM (0.41) KMT2APOLBMEN1
SCHEMBL31535246 0.78 SCN9A (0.50) SCN9A
SCHEMBL22093026 0.77 NR1I2 (0.39) KMT2APOLBMEN1
SCHEMBL517686 0.77 NOTUM (0.47) POLB
SCHEMBL16935559 0.75 KAT2B (0.41) PDE4DPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024118564-A1 CHECKPOINT KINASE 1 (CHK1) INHIBITORS AND USES THEREOF BOUNDLESS BIO, INC. (US) 2024-06-06 WO disclosed