SCHEMBL27281179

SCHEMBL27281179

[CH2]CCNC(=O)c1cc(NC(=O)c2cc(NC(=O)N3CC3)cn2C)cn1C

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 2/20 0.49
HRAS P01112 7/20 0.49
ESR1 P03372 7/20 0.49
ESR2 Q92731 7/20 0.49
KDM4E B2RXH2 3/20 0.48
MAPT P10636 3/20 0.48
POLB P06746 2/20 0.48
HIF1A Q16665 1/20 0.48
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ABL1 P00519 1/20 0.36
RIN1 Q13671 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
FAAH O00519 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27282459 1.00 TOP1 (0.49) TOP1HRASESR1ESR2KDM4E
SCHEMBL27282453 0.92 HRAS (0.48) TOP1HRASESR1ESR2KDM4E
SCHEMBL10693106 0.84 HRAS (0.71) TOP1HRASESR1ESR2KDM4E
SCHEMBL10691121 0.84 HDAC1 (0.55) TOP1HRASESR1ESR2KDM4E
SCHEMBL10691569 0.84 HDAC1 (0.55) TOP1HRASESR1ESR2KDM4E
Hydrochloric Acid SCHEMBL10693753 0.83 KDM4E (0.72) TOP1HRASESR1ESR2KDM4E
Hydrochloric Acid SCHEMBL10693590 0.83 HDAC1 (0.54) TOP1HRASESR1ESR2KDM4E
Hydrochloric Acid SCHEMBL10691977 0.83 HDAC1 (0.54) TOP1HRASESR1ESR2KDM4E
SCHEMBL27272389 0.82 HRAS (0.54) TOP1HRASESR1ESR2KDM4E
SCHEMBL27281879 0.82 HRAS (0.54) TOP1HRASESR1ESR2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1018825-B Process for preparing poly-4-aminopyrrole-2-carboxamido derivatives ERBA FARMITALIA (IT) 1992-10-28 CN disclosed