SCHEMBL27299352

SCHEMBL27299352

COc1ccc(C2(C(=O)O)CC(c3ccccc3)c3ccccc32)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 2/20 0.45
KMT2A Q03164 3/20 0.44
MAPT P10636 2/20 0.44
MEN1 O00255 2/20 0.44
KDM4E B2RXH2 1/20 0.44
EDNRB P24530 1/20 0.43
NPC1 O15118 2/20 0.41
ATM Q13315 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
GAA P10253 1/20 0.41
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
MAPK1 P28482 1/20 0.38
RAB9A P51151 1/20 0.38
KIF11 P52732 1/20 0.37
FFAR1 O14842 1/20 0.37
TSHR P16473 1/20 0.37
RECQL P46063 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27303889 0.93 KMT2A (0.43) EDNRAKMT2AMAPTMEN1KDM4E
SCHEMBL27300785 0.92 MEN1 (0.43) EDNRAKMT2AMAPTMEN1KDM4E
SCHEMBL27296603 0.87 MEN1 (0.47) KMT2AMAPTMEN1KDM4ESLC6A2
SCHEMBL27295612 0.84 DRD1 (0.35) KMT2AMAPTMEN1GAASIGMAR1
SCHEMBL27346085 0.83 GAA (0.39) KMT2AMEN1KDM4EGAASIGMAR1
SCHEMBL14701152 0.80 MEN1 (0.45) EDNRAKMT2AMAPTMEN1KDM4E
SCHEMBL13588376 0.78 KMT2A (0.44) EDNRAKMT2AMAPTMEN1KDM4E
SCHEMBL8304137 0.74 HTR2A (0.46) KMT2AMEN1
SCHEMBL27359306 0.74 HDAC9 (0.55) KMT2AMAPTNPC1SIGMAR1MAPK1
SCHEMBL9543856 0.70 EDNRA (0.46) EDNRAKMT2AMAPTMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1034569-C ET (ENDOTHELIN) receptor antagonists SMITHKLINE BEECHAM CORP (US) 1997-04-16 CN disclosed
CN-1073161-A ET (ENDOTHELIN) receptor antagonists SMITHKLINE BEECHAM CORP (US) 1993-06-16 CN disclosed