SCHEMBL27314717

SCHEMBL27314717

O=C(C(=O)c1cccc2ccccc12)C1=CCCc2c1ccc1c2ccc2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A1 P22736 1/20 0.40
NR4A2 P43354 1/20 0.40
NR4A3 Q92570 1/20 0.40
MMP3 P08254 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
PTPN1 P18031 1/20 0.36
CDC25B P30305 1/20 0.36
PLK1 P53350 1/20 0.36
HPRT1 P00492 1/20 0.36
SOS1 Q07889 2/20 0.36
ALDH1A1 P00352 6/20 0.35
MAPT P10636 5/20 0.35
MEN1 O00255 4/20 0.35
LMNA P02545 4/20 0.35
KMT2A Q03164 4/20 0.35
CYP1A2 P05177 3/20 0.35
HPGD P15428 3/20 0.35
MAPK1 P28482 3/20 0.35
POLB P06746 3/20 0.35
NPSR1 Q6W5P4 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7218991 0.72 NR4A1 (0.71) NR4A1NR4A2NR4A3MMP3HDAC8
SCHEMBL29494693 0.72 NR4A1 (0.71) NR4A1NR4A2NR4A3MMP3HDAC8
SCHEMBL27523850 0.71 HPRT1 (0.41) HPRT1ALDH1A1MAPTMEN1LMNA
SCHEMBL15903547 0.71 HPRT1 (0.44) NR4A1NR4A2NR4A3HPRT1SOS1
SCHEMBL15903797 0.69 HPRT1 (0.41) HPRT1SOS1ALDH1A1MAPTMEN1
SCHEMBL31464018 0.69 ALDH1A1 (0.46) HPRT1SOS1ALDH1A1MAPTMEN1
SCHEMBL28513228 0.68 NR4A1 (0.55) NR4A1NR4A2NR4A3MMP3HDAC8
SCHEMBL548063 0.68 NR4A1 (0.55) NR4A1NR4A2NR4A3MMP3HDAC8
SCHEMBL14211980 0.67 NR4A1 (0.64) NR4A1NR4A2NR4A3MMP3HDAC8
SCHEMBL1314383 0.67 HPRT1 (0.56) NR4A1NR4A2NR4A3MMP3HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1030986-C Pyrrolopyrazine HOFFMANN LA ROCHE (CH) 1996-02-14 CN disclosed