SCHEMBL273173

SCHEMBL273173

Cc1cc(C)c2c(n1)sc1c(=O)[nH]cnc12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 4/20 0.57
KDM4E B2RXH2 5/20 0.55
HPGD P15428 4/20 0.55
ALDH1A1 P00352 4/20 0.55
MAPT P10636 4/20 0.55
PIM1 P11309 2/20 0.55
PRKACA P17612 2/20 0.55
GSK3A P49840 2/20 0.55
DYRK1A Q13627 2/20 0.55
CDC7 O00311 1/20 0.55
PLK4 O00444 1/20 0.55
IKBKB O14920 1/20 0.55
AURKA O14965 1/20 0.55
CHUK O15111 1/20 0.55
ROCK2 O75116 1/20 0.55
FYN P06241 1/20 0.55
RPS6KB1 P23443 1/20 0.55
CDK2 P24941 1/20 0.55
MARK3 P27448 1/20 0.55
AKT1 P31749 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30410968 0.92 CDC7 (0.51) CHRM4KDM4EHPGDALDH1A1MAPT
SCHEMBL18666379 0.87 HPGD (0.53) CHRM4KDM4EHPGDALDH1A1MAPT
SCHEMBL432011 0.78 KDM4E (0.67) CHRM4KDM4EHPGDALDH1A1MAPT
SCHEMBL5992997 0.78 KDM4E (0.56) CHRM4KDM4EHPGDALDH1A1MAPT
SCHEMBL278791 0.73 POLB (0.65) CHRM4KDM4EALDH1A1MAPTPIM1
SCHEMBL21523008 0.73 CHRM4 (1.00) CHRM4KDM4EALDH1A1MAPTPIM1
SCHEMBL23273359 0.72 PARP1 (0.54) KDM4EHPGDALDH1A1PIM1GAA
SCHEMBL4903009 0.71 CDC7 (1.00) CHRM4KDM4EHPGDALDH1A1MAPT
SCHEMBL4207656 0.71 PARP1 (0.54) KDM4EHPGDALDH1A1MAPTPIM1
SCHEMBL30989229 0.71 KDM4E (0.66) CHRM4KDM4EHPGDALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4172361-A1 DETECTION OF METHYLATION STATUS Pentabase APS (DK) 2023-05-03 EP claimed
WO-2022002958-A1 DETECTION OF METHYLATION STATUS PENTABASE APS (DK) 2022-01-06 WO claimed
US-10988810-B2 Methods and materials for detection of mutations PENTABASE APS (DK) 2021-04-27 US claimed
US-20190085400-A1 METHODS AND MATERIALS FOR DETECTION OF MUTATIONS PENTABASE APS (DK) 2019-03-21 US claimed
EP-3350347-A1 METHODS AND MATERIALS FOR DETECTION OF MUTATIONS Pentabase APS (DK) 2018-07-25 EP claimed
WO-2017045689-A1 METHODS AND MATERIALS FOR DETECTION OF MUTATIONS PENTABASE APS (DK) 2017-03-23 WO claimed
EP-2004847-A2 OLIGONUCLEOTIDES COMPRISING SIGNALLING PAIRS AND HYDROPHOBIC NUCLEOTIDES, STEMLESS BEACONS, FOR DETECTION OF NUCLEIC ACIDS, METHYLATION STATUS AND MUTANTS OF NUCLEIC ACIDS Pentabase Aps (DK) 2008-12-24 EP claimed
WO-2007104318-A2 OLIGONUCLEOTIDES COMPRISING SIGNALLING PAIRS AND HYDROPHOBIC NUCLEOTIDES, STEMLESS BEACONS, FOR DETECTION OF NUCLEIC ACIDS, METHYLATION STATUS AND MUTANTS OF NUCLEIC ACIDS PENTABASE APS (DK) 2007-09-20 WO claimed
US-20250346955-A1 DETECTION OF METHYLATION STATUS PENTABASE APS (DK) 2025-11-13 US disclosed
EP-4172361-B1 DETECTION OF METHYLATION STATUS PENTABASE AS (DK) 2024-08-07 EP disclosed
EP-4172361-A1 DETECTION OF METHYLATION STATUS Pentabase APS (DK) 2023-05-03 EP disclosed
US-20220205024-A1 MELTING TEMPERATURE METHODS, KITS AND REPORTER OLIGO FOR DETECTING VARIANT NUCLEIC ACIDS PENTABASE APS (DK) 2022-06-30 US disclosed
WO-2022002958-A1 DETECTION OF METHYLATION STATUS PENTABASE APS (DK) 2022-01-06 WO disclosed
US-10988810-B2 Methods and materials for detection of mutations PENTABASE APS (DK) 2021-04-27 US disclosed
US-20100068704-A1 OLIGONUCLEOTIDES COMPRISING SIGNALLING PAIRS AND HYDROPHOBIC NUCLEOTIDES, STEMLESS BEACONS, FOR DETECTION OF NUCLEIC ACIDS, METHYLATION STATUS AND MUTANTS OF NUCLEIC ACIDS PENTABASE APS (DK) 2010-03-18 US disclosed
US-20100068704-A1 OLIGONUCLEOTIDES COMPRISING SIGNALLING PAIRS AND HYDROPHOBIC NUCLEOTIDES, STEMLESS BEACONS, FOR DETECTION OF NUCLEIC ACIDS, METHYLATION STATUS AND MUTANTS OF NUCLEIC ACIDS PENTABASE APS (DK) 2010-03-18 US disclosed
US-20100068704-A1 OLIGONUCLEOTIDES COMPRISING SIGNALLING PAIRS AND HYDROPHOBIC NUCLEOTIDES, STEMLESS BEACONS, FOR DETECTION OF NUCLEIC ACIDS, METHYLATION STATUS AND MUTANTS OF NUCLEIC ACIDS PENTABASE APS (DK) 2010-03-18 US disclosed
EP-2004847-A2 OLIGONUCLEOTIDES COMPRISING SIGNALLING PAIRS AND HYDROPHOBIC NUCLEOTIDES, STEMLESS BEACONS, FOR DETECTION OF NUCLEIC ACIDS, METHYLATION STATUS AND MUTANTS OF NUCLEIC ACIDS Pentabase Aps (DK) 2008-12-24 EP disclosed
WO-2007104318-A2 OLIGONUCLEOTIDES COMPRISING SIGNALLING PAIRS AND HYDROPHOBIC NUCLEOTIDES, STEMLESS BEACONS, FOR DETECTION OF NUCLEIC ACIDS, METHYLATION STATUS AND MUTANTS OF NUCLEIC ACIDS PENTABASE APS (DK) 2007-09-20 WO disclosed
WO-2007104318-A2 OLIGONUCLEOTIDES COMPRISING SIGNALLING PAIRS AND HYDROPHOBIC NUCLEOTIDES, STEMLESS BEACONS, FOR DETECTION OF NUCLEIC ACIDS, METHYLATION STATUS AND MUTANTS OF NUCLEIC ACIDS PENTABASE APS (DK) 2007-09-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100068704-A1 OLIGONUCLEOTIDES COMPRISING SIGNALLING PAIRS AND HYDROPHOBIC NUCLEOTIDES, STEMLESS BEACONS, FOR DETECTION OF NUCLEIC ACIDS, METHYLATION STATUS AND MUTANTS OF NUCLEIC ACIDS DNMT1, DNMT3A, DNMT3L CHRM4 2985/4885KDM4E 4552/4885HPGD 3576/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.