SCHEMBL2732891

SCHEMBL2732891

CN(Cc1ccccc1)C1COCCN(C(=O)O)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.46
JAK2 O60674 1/20 0.45
JAK1 P23458 1/20 0.45
FKBP1A P62942 1/20 0.43
OPRM1 P35372 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
HDAC1 Q13547 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
AGTR2 P50052 2/20 0.42
LTA4H P09960 1/20 0.41
MEN1 O00255 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
RORC P51449 1/20 0.41
CACNA1G O43497 1/20 0.40
CACNA1H O95180 1/20 0.40
CACNA1I Q9P0X4 1/20 0.40
MCHR1 Q99705 1/20 0.40
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2732226 0.85 JAK2 (0.65) KMT2AJAK2JAK1MEN1NPSR1
SCHEMBL18424508 0.83 KMT2A (0.56) KMT2AJAK2JAK1OPRM1SIGMAR1
SCHEMBL144125 0.82 KMT2A (0.51) KMT2AJAK2JAK1OPRM1SIGMAR1
SCHEMBL785972 0.77 JAK2 (0.54) KMT2AJAK2JAK1OPRM1SIGMAR1
SCHEMBL2731227 0.76 KMT2A (0.44) KMT2AJAK2JAK1OPRM1SIGMAR1
SCHEMBL16192363 0.75 JAK2 (0.74) KMT2AJAK2JAK1OPRM1SIGMAR1
SCHEMBL28568037 0.75 JAK2 (0.64) KMT2AJAK2JAK1OPRM1SIGMAR1
SCHEMBL28568035 0.75 JAK2 (0.64) KMT2AJAK2JAK1OPRM1SIGMAR1
SCHEMBL17274372 0.75 NAAA (0.63) KMT2AJAK2JAK1HDAC1MCHR1
SCHEMBL13132647 0.74 GRIN2B (0.49) KMT2AOPRM1SIGMAR1HDAC1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2632898-A1 HETEROCYCLIC TYROSINE KINASE INHIBITORS Biogen Idec MA Inc. (US) 2013-09-04 EP disclosed
WO-2012058645-A1 HETEROCYCLIC TYROSINE KINASE INHIBITORS BIOGEN IDEC MA INC. (US) 2012-05-03 WO disclosed