SCHEMBL2733404

SCHEMBL2733404

Cc1cccc(N(C(N)=O)c2ccc(-c3cccc4c3CNC4=O)c(F)c2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 19/20 0.59
ROCK2 O75116 5/20 0.44
AURKB Q96GD4 5/20 0.44
EPHA2 P29317 4/20 0.44
FLT4 P35916 4/20 0.44
FLT3 P36888 4/20 0.44
RPS6KB1 P23443 4/20 0.44
ROCK1 Q13464 4/20 0.44
TAOK1 Q7L7X3 4/20 0.44
HIPK4 Q8NE63 4/20 0.44
RET P07949 4/20 0.44
PLK4 O00444 3/20 0.44
NTRK1 P04629 3/20 0.44
MET P08581 3/20 0.44
NTRK2 Q16620 3/20 0.44
ALK Q9UM73 3/20 0.44
FLT1 P17948 3/20 0.44
MAP4K4 O95819 3/20 0.44
LCK P06239 3/20 0.44
BLK P51451 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5794432 0.86 KDR (0.63) KDRROCK2AURKBEPHA2FLT4
SCHEMBL5880331 0.83 KDR (0.55) KDRROCK2AURKBEPHA2FLT4
SCHEMBL5750826 0.78 KDR (0.51) KDRROCK2AURKBEPHA2FLT4
SCHEMBL2732814 0.78 KDR (0.56) KDRROCK2AURKBEPHA2FLT4
SCHEMBL2733951 0.77 KDR (0.55) KDRROCK2AURKBEPHA2FLT4
SCHEMBL2732944 0.76 KDR (0.58) KDRROCK2AURKBEPHA2FLT4
SCHEMBL5745576 0.75 KDR (0.44) KDRROCK2AURKBEPHA2FLT4
SCHEMBL5880323 0.75 KDR (0.49) KDRROCK2AURKBEPHA2FLT4
SCHEMBL5880325 0.75 KDR (0.50) KDRROCK2AURKBEPHA2FLT4
SCHEMBL1334456 0.74 KDR (1.00) KDRROCK2AURKBEPHA2FLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012061602-A1 ISOINDOLINONE KINASE INHIBITORS ABBOTT LABORATORIES (US) 2012-05-10 WO disclosed