SCHEMBL27358558

SCHEMBL27358558

C[C@@H]1CCC(C#N)N1C(=O)OC(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 11/20 0.48
CHRM2 P08172 1/20 0.45
CHRM1 P11229 1/20 0.45
CHRM3 P20309 1/20 0.45
CTSK P43235 1/20 0.40
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
HPGD P15428 1/20 0.38
PREP P48147 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18501444 1.00 DPP4 (0.48) DPP4CHRM2CHRM1CHRM3CTSK
SCHEMBL25505419 0.84 CHRM2 (0.45) DPP4CHRM2CHRM1CHRM3MEN1
SCHEMBL26782299 0.84 CHRM2 (0.45) DPP4CHRM2CHRM1CHRM3MEN1
SCHEMBL29102351 0.84 CHRM2 (0.45) DPP4CHRM2CHRM1CHRM3MEN1
SCHEMBL26782288 0.84 CHRM2 (0.45) DPP4CHRM2CHRM1CHRM3MEN1
SCHEMBL18901924 0.84 CHRM2 (0.45) DPP4CHRM2CHRM1CHRM3MEN1
SCHEMBL18901834 0.84 CHRM2 (0.45) DPP4CHRM2CHRM1CHRM3MEN1
SCHEMBL21441814 0.82 CHRM2 (0.56) CHRM2CHRM1CHRM3HPGDPREP
SCHEMBL12333780 0.82 CHRM2 (0.56) CHRM2CHRM1CHRM3HPGDPREP
SCHEMBL880528 0.82 CHRM2 (0.56) CHRM2CHRM1CHRM3HPGDPREP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024091409-A1 TRICYCLIC DERIVATIVES AS KRAS INHIBITORS NIKANG THERAPEUTICS, INC. (US) 2024-05-02 WO disclosed
WO-2024050742-A1 BIFUNCTIONAL COMPOUNDS FOR DEGRADING KRAS G12D VIA UBIQUITIN PROTEASOME PATHWAY NIKANG THERAPEUTICS, INC. (US) 2024-03-14 WO disclosed