SCHEMBL27366276

SCHEMBL27366276

CCCCc1ccc(C(F)(F)F)cc1C(=O)OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.54
PLK1 P53350 1/20 0.45
RXRA P19793 5/20 0.44
NR1H2 P55055 5/20 0.44
PPARG P37231 2/20 0.44
PPARD Q03181 2/20 0.44
PPARA Q07869 2/20 0.44
MRGPRX4 Q96LA9 1/20 0.44
CNR2 P34972 2/20 0.43
CES2 O00748 1/20 0.43
CNR1 P21554 1/20 0.43
NR1H3 Q13133 3/20 0.42
NOTUM Q6P988 1/20 0.41
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ESRRA P11474 1/20 0.40
LIPC P11150 1/20 0.39
LIPG Q9Y5X9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8612829 0.89 CFTR (0.46) CFTRPLK1RXRANR1H2PPARG
SCHEMBL13730307 0.87 CFTR (0.60) CFTRRXRANR1H2MRGPRX4CES2
Ammonia Solution, Strong SCHEMBL7107044 0.83 PLK1 (0.52) PLK1RXRANR1H2PPARDPPARA
SCHEMBL477875 0.82 CFTR (0.59) CFTRRXRANR1H2MRGPRX4CES2
SCHEMBL22826631 0.81 TYR (0.42) CNR2CNR1KDM4EALDH1A1SMN1; SMN2
SCHEMBL1435026 0.81 CFTR (0.57) CFTRRXRANR1H2MRGPRX4CES2
SCHEMBL8612587 0.80 CFTR (0.48) CFTRRXRANR1H2PPARGPPARD
SCHEMBL2358405 0.79 PLK1 (0.51) PLK1RXRANR1H2CNR2CES2
SCHEMBL4107553 0.79 CFTR (0.55) CFTRRXRANR1H2MRGPRX4CES2
Ammonia Solution, Strong SCHEMBL27818289 0.78 KDM4E (0.51) PLK1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1064955-C Fluorine-containing benzoylguanidines MERCK PATENT GMBH (DE) 2001-04-25 CN disclosed
CN-1143632-A Fluorine-containing benzoylguanidines MERCK PATENT GMBH (DE) 1997-02-26 CN disclosed