SCHEMBL27378784

SCHEMBL27378784

COC(=O)[C@H]1C[C@@H]1c1cncc(-n2c(=O)[nH]c3cc(-c4ccccc4Cl)sc3c2=O)c1C

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ERCC5 P28715 1/20 0.32
FEN1 P39748 1/20 0.32
EGLN3 Q9H6Z9 1/20 0.31
CHEK1 O14757 1/20 0.31
TSHR P16473 1/20 0.30
ADRA1B P35368 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29326549 0.90 HSD17B10 (0.38) ALDH1A1MEN1RAB9AKMT2AHSD17B10
SCHEMBL27378764 0.85 TNKS2 (0.39) ALDH1A1MEN1RAB9AKMT2AHSD17B10
SCHEMBL27381086 0.84 ERCC5 (0.34) ERCC5FEN1CHEK1ADRA1B
SCHEMBL27192121 0.80 MAPK14 (0.33) ERCC5FEN1
SCHEMBL30701990 0.80 MAPK14 (0.33) ERCC5FEN1
SCHEMBL27378775 0.80 ERCC5 (0.38) ALDH1A1MEN1KMT2AERCC5FEN1
SCHEMBL27192043 0.79 ERCC5 (0.36) ALDH1A1MEN1KMT2AERCC5FEN1
SCHEMBL30702084 0.79 ERCC5 (0.36) ALDH1A1MEN1KMT2AERCC5FEN1
SCHEMBL27379530 0.77 TNKS2 (0.35) ALDH1A1MEN1KMT2AHSD17B10ERCC5
SCHEMBL27381102 0.75 MAP4K1 (0.33) HSD17B10ERCC5FEN1EGLN3CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024031089-A1 SARS-COV2 MAIN PROTEASE INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-08 WO disclosed