SCHEMBL27388252

SCHEMBL27388252

N[C@@H](Cc1ccc(O)cc1)C(=O)N1CC[CH]CC1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 6/20 0.63
DPP4 P27487 5/20 0.54
SLC7A5 Q01650 1/20 0.54
OPRD1 P41143 1/20 0.52
HRH2 P25021 1/20 0.48
HRH1 P35367 1/20 0.48
SMYD3 Q9H7B4 1/20 0.48
ARG1 P05089 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14390395 0.88 HDAC8 (0.67) HDAC8DPP4SLC7A5OPRD1HRH2
SCHEMBL5746200 0.84 HDAC8 (0.62) HDAC8DPP4SLC7A5OPRD1HRH2
SCHEMBL5746194 0.84 HDAC8 (0.62) HDAC8DPP4SLC7A5OPRD1HRH2
Hydrochloric Acid SCHEMBL6165142 0.81 HDAC8 (0.61) HDAC8DPP4SLC7A5OPRD1HRH2
Hydrochloric Acid SCHEMBL6165132 0.81 HDAC8 (0.61) HDAC8DPP4SLC7A5OPRD1HRH2
Trifluoroacetic Acid SCHEMBL6824509 0.80 HDAC8 (0.58) HDAC8DPP4SLC7A5OPRD1HRH2
SCHEMBL7363744 0.79 OPRD1 (0.61) HDAC8DPP4SLC7A5OPRD1HRH2
SCHEMBL30429936 0.78 DPP4 (0.60) HDAC8DPP4SLC7A5OPRD1HRH2
SCHEMBL7360569 0.78 HDAC8 (0.55) HDAC8DPP4SLC7A5OPRD1HRH2
SCHEMBL4776727 0.78 HDAC8 (1.00) HDAC8DPP4SLC7A5OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1075062-C Acetic acid derivatives HOFFMANN LA ROCHE (CH) 2001-11-21 CN disclosed
CN-1209063-A Vitronection receptor antagonists SMITHKLINE BEECHAM CORP (US) 1999-02-24 CN disclosed
CN-1209060-A Vitronectin receptor antagonists SMITHKLINE BEECHAM CORP (US) 1999-02-24 CN disclosed
CN-1112104-A Acetic acid derivatives HOFFMANN LA ROCHE (CH) 1995-11-22 CN disclosed