SCHEMBL27399207

SCHEMBL27399207

Cn1c(OC=O)c(-c2ccc(F)cc2)c2ccsc2c1=O

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.35
PKLR P30613 1/20 0.35
MAPK14 Q16539 1/20 0.34
PTGS1 P23219 3/20 0.34
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32
MAPT P10636 1/20 0.32
PTGS2 P35354 2/20 0.32
DPP4 P27487 1/20 0.32
RXFP1 Q9HBX9 2/20 0.31
NEK1 Q96PY6 1/20 0.31
CENPE Q02224 2/20 0.31
BRD4 O60885 1/20 0.31
NR1D1 P20393 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
SLC11A2 P49281 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7850622 0.75 GRIA2 (0.44) PKMPKLRMAPK14PTGS1RXFP1
SCHEMBL7852329 0.72 TP53 (0.41) PKMTSHRHTTMAPTCENPE
SCHEMBL7850615 0.68 GRIA2 (0.44) PKMPKLRMAPK14PTGS1NEK1
SCHEMBL7849856 0.67 TACR1 (0.66) TSHRHTTMAPTRXFP1
SCHEMBL7843050 0.62 SLC11A2 (0.43) PKMHTTSLC11A2
SCHEMBL13641556 0.60 ADORA1 (0.41) PKMHTT
SCHEMBL7852458 0.59 TSHR (0.49) TSHRHTTMAPTSLC11A2
SCHEMBL17290337 0.59 SLC11A2 (0.55) MAPK14HTTMAPTSLC11A2
SCHEMBL2553123 0.58 GPR3 (0.50) HTTMAPTRXFP1
SCHEMBL19661324 0.58 TSHR (0.36) TSHRMAPTBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1052004-C Heterocyclic compounds, their production and use TALCEDA CHEMICAL IND LTD (JP) 2000-05-03 CN disclosed
CN-1107476-A Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-08-30 CN disclosed