SCHEMBL27426751

SCHEMBL27426751

CSc1ccc(C(Cc2ccccc2)C(C)=O)cc1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.57
ESR2 Q92731 1/20 0.57
EPHX1 P07099 1/20 0.50
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
CHRM1 P11229 5/20 0.44
RAB9A P51151 2/20 0.44
UBE2N P61088 1/20 0.44
NPC1 O15118 1/20 0.44
MAPT P10636 1/20 0.44
KDM4E B2RXH2 1/20 0.43
SLC6A4 P31645 2/20 0.42
ALPI P09923 1/20 0.42
PKM P14618 1/20 0.42
PTGS1 P23219 1/20 0.42
XIAP P98170 1/20 0.42
SLC7A5 Q01650 1/20 0.42
ACACB O00763 1/20 0.42
P4HTM Q9NXG6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27426752 0.94 ESR1 (0.57) ESR1ESR2EPHX1MEN1KMT2A
SCHEMBL5272849 0.85 EPHX1 (0.67) ESR1ESR2EPHX1CHRM1RAB9A
SCHEMBL27667714 0.82 ESR1 (0.83) ESR1ESR2EPHX1CHRM1UBE2N
SCHEMBL7042498 0.78 SLC6A4 (0.48) MEN1KMT2ARAB9ANPC1MAPT
SCHEMBL13243493 0.78 PPARG (0.57) ESR1ESR2EPHX1MEN1KMT2A
SCHEMBL28287871 0.78 SLC6A2 (0.56) ESR1ESR2EPHX1MEN1KMT2A
SCHEMBL27403469 0.77 ESR1 (0.55) ESR1ESR2EPHX1CHRM1UBE2N
SCHEMBL27581400 0.76 NPC1 (0.54) ESR1ESR2EPHX1MEN1KMT2A
SCHEMBL28980645 0.76 MEN1 (0.49) MEN1KMT2ARAB9ANPC1MAPT
SCHEMBL6049128 0.76 ESR1 (0.83) ESR1ESR2EPHX1CHRM1UBE2N

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1214790-C Medicinal composition for treating inflammation SEARLE & CO (US) 2005-08-17 CN disclosed
CN-1442139-A Medicinal composition for treating inflammation SEARLE & CO (US) 2003-09-17 CN disclosed
CN-1107058-C Substituted isoxazoles for the treatment of disorders SEARLE & CO (US) 2003-04-30 CN disclosed
CN-1181075-A Substituted isoxazoles for the treatment of disorders SEARLE & CO (US) 1998-05-06 CN disclosed