SCHEMBL27426752

SCHEMBL27426752

CSc1ccc(CC(C(C)=O)c2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.57
ESR2 Q92731 1/20 0.57
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
EPHX1 P07099 1/20 0.50
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
SLC6A4 P31645 6/20 0.46
MAOA P21397 1/20 0.45
SLC6A2 P23975 1/20 0.45
SLC6A3 Q01959 1/20 0.45
ACACB O00763 1/20 0.45
CHRM1 P11229 4/20 0.44
UBE2N P61088 1/20 0.44
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27426751 0.94 ESR1 (0.57) ESR1ESR2MEN1KMT2AEPHX1
SCHEMBL5272849 0.85 EPHX1 (0.67) ESR1ESR2EPHX1CHRM1UBE2N
SCHEMBL3371227 0.82 ESR1 (0.62) ESR1ESR2MEN1KMT2AEPHX1
SCHEMBL6049128 0.82 ESR1 (0.83) ESR1ESR2EPHX1LMNACHRM1
SCHEMBL3371208 0.81 ESR1 (0.60) ESR1ESR2EPHX1CHRM1UBE2N
SCHEMBL6958211 0.81 ESR1 (0.60) ESR1ESR2EPHX1ALDH1A1CHRM1
SCHEMBL3368827 0.77 ESR1 (0.55) ESR1ESR2EPHX1CHRM1UBE2N
SCHEMBL27581401 0.76 ESR1 (0.54) ESR1ESR2MEN1KMT2AEPHX1
SCHEMBL28980645 0.76 MEN1 (0.49) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL27667714 0.76 ESR1 (0.83) ESR1ESR2EPHX1LMNACHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1214790-C Medicinal composition for treating inflammation SEARLE & CO (US) 2005-08-17 CN disclosed
CN-1442139-A Medicinal composition for treating inflammation SEARLE & CO (US) 2003-09-17 CN disclosed
CN-1107058-C Substituted isoxazoles for the treatment of disorders SEARLE & CO (US) 2003-04-30 CN disclosed
CN-1181075-A Substituted isoxazoles for the treatment of disorders SEARLE & CO (US) 1998-05-06 CN disclosed