SCHEMBL27427552

SCHEMBL27427552

N=C(NCc1ccccc1)NC(=O)c1cc2ccccc2[nH]1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.56
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
CA9 Q16790 1/20 0.56
KDM4E B2RXH2 4/20 0.56
ALDH1A1 P00352 2/20 0.56
GAA P10253 1/20 0.56
MAPK1 P28482 1/20 0.56
IDO1 P14902 1/20 0.53
NPC1 O15118 1/20 0.53
LMNA P02545 1/20 0.53
RAB9A P51151 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
HDAC2 Q92769 2/20 0.52
HDAC3 O15379 1/20 0.52
HDAC1 Q13547 1/20 0.52
NCOR2 Q9Y618 1/20 0.52
DRD2 P14416 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8689817 0.99 CA12 (0.55) CA12CA1CA2CA9KDM4E
SCHEMBL2735969 0.86 CA12 (0.72) CA12CA1CA2CA9KDM4E
SCHEMBL7877575 0.80 KDM4E (0.59) KDM4EALDH1A1GAAMAPK1NPC1
Hydrochloric Acid SCHEMBL3926581 0.80 IDO1 (0.52) CA12CA1CA2CA9KDM4E
Hydrochloric Acid SCHEMBL7882333 0.79 KDM4E (0.57) KDM4EALDH1A1GAAMAPK1NPC1
SCHEMBL8227820 0.78 ITGB3 (0.69) CA12CA1CA2CA9KDM4E
SCHEMBL13587037 0.78 HDAC2 (0.67) CA12CA1CA2CA9KDM4E
SCHEMBL6657027 0.77 HDAC2 (0.67) CA12CA1CA2CA9KDM4E
SCHEMBL14269112 0.77 IDO1 (0.65) KDM4EALDH1A1GAAMAPK1IDO1
SCHEMBL1952751 0.76 KDM4E (0.67) KDM4EALDH1A1GAAMAPK1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1136038-A Indoloylguanidine derivatives SUMITOMO PHARMACEUTICS K K (JP) 1996-11-20 CN disclosed
CN-1106800-A Indoloylguanidine derivatives SUMITOMO PHARMA (JP) 1995-08-16 CN disclosed