SCHEMBL27428191

SCHEMBL27428191

[c]1nc2ccc(-c3nccs3)cc2[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.41
ADRB2 P07550 1/20 0.39
CYP2A6 P11509 1/20 0.38
TLR8 Q9NR97 2/20 0.37
TLR7 Q9NYK1 2/20 0.37
QPCT Q16769 1/20 0.36
LRRK2 Q5S007 1/20 0.36
PDE10A Q9Y233 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
CHEK1 O14757 1/20 0.35
SMPD3 Q9NY59 1/20 0.35
HDAC2 Q92769 1/20 0.34
METAP1 P53582 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
VCP P55072 1/20 0.34
TLR9 Q9NR96 1/20 0.33
CHEK2 O96017 1/20 0.33
ESR1 P03372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8094750 0.88 PDPK1 (0.42) PDPK1LOXL2ADRB2CYP2A6TLR8
SCHEMBL8499706 0.72 PDE10A (0.44) PDPK1LOXL2ADRB2CYP2A6TLR8
SCHEMBL8088436 0.72 PDE10A (0.44) PDPK1LOXL2ADRB2CYP2A6TLR8
SCHEMBL27947333 0.70 FGFR1 (0.43) QPCTCHEK1
SCHEMBL722198 0.70 PDPK1 (0.77) PDPK1LOXL2ADRB2CYP2A6PTGDR2
SCHEMBL27947326 0.69 MAP4K4 (0.39) PDPK1QPCTCHEK1CHEK2
SCHEMBL13142475 0.69 PDPK1 (0.57) PDPK1LOXL2ADRB2CYP2A6PTGDR2
SCHEMBL28151600 0.69 PDPK1 (0.44) PDPK1LOXL2ADRB2CYP2A6TLR8
SCHEMBL26259866 0.68 PDPK1 (0.55) PDPK1LOXL2ADRB2CYP2A6TLR8
SCHEMBL15805858 0.67 PDPK1 (0.72) PDPK1LOXL2ADRB2CYP2A6PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1105720-C Imidazopyridazines compound AOTANNA MEDICINE AG (DE) 2003-04-16 CN disclosed
CN-1246120-A Imidazopyridazines compound BYK GULDEN LOMBERG CHEM FAB (DE) 2000-03-01 CN disclosed