SCHEMBL8499706

SCHEMBL8499706

Clc1nc2ccc(-c3nccs3)cc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.44
PDPK1 O15530 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.41
METAP1 P53582 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
TLR8 Q9NR97 1/20 0.39
TLR7 Q9NYK1 1/20 0.39
ADRB2 P07550 1/20 0.38
PRKAG1 P54619 1/20 0.38
PRKAA2 P54646 1/20 0.38
PRKAB1 Q9Y478 1/20 0.38
CYP2A6 P11509 1/20 0.37
NPC1 O15118 3/20 0.37
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 2/20 0.36
ALDH1A1 P00352 2/20 0.36
TP53 P04637 2/20 0.36
GAA P10253 2/20 0.36
MAPT P10636 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8499704 0.88 TLR8 (0.41) PDE10APDPK1LOXL2METAP1ADORA2A
SCHEMBL8088436 0.82 PDE10A (0.44) PDE10APDPK1LOXL2METAP1TLR8
SCHEMBL27428191 0.72 PDPK1 (0.42) PDE10APDPK1LOXL2METAP1ADORA2A
SCHEMBL13142475 0.71 PDPK1 (0.57) PDPK1LOXL2METAP1ADORA2AADORA1
SCHEMBL2878859 0.71 KDM4E (0.54) PDE10ANPC1KDM4EMEN1ALDH1A1
SCHEMBL28151600 0.71 PDPK1 (0.44) PDPK1LOXL2METAP1ADORA2AADORA1
SCHEMBL679566 0.71 PDPK1 (0.52) PDPK1LOXL2ADORA2AADORA1ADRB2
SCHEMBL8501749 0.71 TLR8 (0.46) PDE10APDPK1LOXL2METAP1TLR8
SCHEMBL8501746 0.71 TLR8 (0.41) PDE10APDPK1LOXL2METAP1ADORA2A
SCHEMBL26259866 0.70 PDPK1 (0.55) PDPK1LOXL2METAP1ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946559-A2 IMIDAZOPYRIDAZINES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1999-10-06 EP disclosed
WO-1998028299-A2 IMIDAZOPYRIDAZINES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1998-07-02 WO disclosed