SCHEMBL27439600

SCHEMBL27439600

NC(OCc1ccccc1)c1c[c]ccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.42
SLC6A4 P31645 2/20 0.42
SLC6A3 Q01959 2/20 0.42
TACR1 P25103 3/20 0.41
SLC1A3 P43003 2/20 0.41
SLC1A2 P43004 2/20 0.41
SLC1A1 P43005 2/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
IDO1 P14902 1/20 0.37
AGXT P21549 1/20 0.36
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
AOC3 Q16853 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9117050 0.82 TACR1 (0.52) SLC6A2SLC6A4SLC6A3TACR1SLC1A3
SCHEMBL27443072 0.81 SLC1A3 (0.44) SLC6A2SLC6A4SLC6A3TACR1SLC1A3
SCHEMBL8333871 0.81 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3TACR1SLC1A3
SCHEMBL27481651 0.80 SLC1A3 (0.42) SLC6A2SLC6A4SLC6A3TACR1SLC1A3
SCHEMBL8338564 0.77 TACR1 (0.45) SLC6A2SLC6A4SLC6A3TACR1SLC1A1
SCHEMBL27928229 0.75 SLC6A2 (0.31) SLC6A2SLC6A4SLC6A3
SCHEMBL27710223 0.72 ALDH1A1 (0.41) KMT2AMEN1TSHRSMN1; SMN2
SCHEMBL7013321 0.71 GRIN2D (0.42) SLC6A2SLC6A4SLC6A3CYP1A2CYP2D6
SCHEMBL6753036 0.71 GRIN2D (0.42) SLC6A2SLC6A4SLC6A3CYP1A2CYP2D6
SCHEMBL992838 0.71 IDO1 (0.47) SLC6A2SLC6A4SLC6A3TACR1SLC1A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1122033-C Triazolopurine derivatives, pharmaceutical compositions containing the same OTSUKE PHARMACEUTICAL FACTORY (JP) 2003-09-24 CN disclosed
CN-1301266-A Triazolopurine derivatives, pharmaceutical composition containing the same, adenosine A3 receptor affinity agent, and asthma therapeutic agent OTSUKA PHARMACEUITCAL FACTORY (JP) 2001-06-27 CN disclosed