SCHEMBL27445552

SCHEMBL27445552

CCCc1ccc2c(c1)CCCNC2=O

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP11 Q9NR21 9/20 0.52
PARP10 Q53GL7 9/20 0.49
HTR2C P28335 2/20 0.43
HTR2B P41595 2/20 0.43
HTR2A P28223 1/20 0.43
GSK3B P49841 1/20 0.41
GRM5 P41594 6/20 0.40
PARP1 P09874 2/20 0.39
PDPK1 O15530 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27446376 0.88 PARP11 (0.55) PARP11PARP10HTR2CHTR2BHTR2A
SCHEMBL19838605 0.82 PARP11 (0.55) PARP11PARP10GSK3BGRM5PARP1
SCHEMBL19852063 0.81 PARP11 (0.51) PARP11PARP10GSK3BPARP1
SCHEMBL8255407 0.79 PARP10 (0.59) PARP11PARP10HTR2CHTR2BHTR2A
SCHEMBL10911695 0.78 KDM4E (0.55) HTR2CHTR2BHTR2A
SCHEMBL10168733 0.78 PARP11 (0.66) PARP11PARP10GRM5PARP1PDPK1
SCHEMBL23777279 0.78 PARP11 (0.55) PARP11PARP10GSK3BGRM5
SCHEMBL12090727 0.76 PARP10 (0.81) PARP11PARP10GSK3BGRM5PARP1
SCHEMBL23160638 0.75 PARP1 (0.49) PARP11PARP10GSK3BGRM5PARP1
SCHEMBL19386434 0.75 PARP11 (0.61) PARP11PARP10GRM5PARP1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024119122-A1 CDK INHIBITORS AND METHODS AND USE THEREOF RELAY THERAPEUTICS, INC. (US) 2024-06-06 WO disclosed