SCHEMBL27459795

SCHEMBL27459795

Cc1cc2c(Nc3ccc(Br)c(F)c3)ncnc2cn1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 12/20 0.53
GRM1 Q13255 1/20 0.51
ERBB2 P04626 3/20 0.51
HDAC1 Q13547 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
TNK2 Q07912 1/20 0.48
MKNK1 Q9BUB5 1/20 0.48
MAPK1 P28482 1/20 0.46
PIP4K2A P48426 1/20 0.46
ERBB4 Q15303 1/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7535181 0.99 EGFR (0.52) EGFRGRM1ERBB2HDAC1HDAC6
SCHEMBL7661721 0.85 GRM1 (0.56) EGFRGRM1ERBB2MEN1KMT2A
Hydrochloric Acid SCHEMBL7536080 0.84 GRM1 (0.55) EGFRGRM1ERBB2MEN1KMT2A
SCHEMBL7543155 0.82 GRM1 (0.74) EGFRGRM1ERBB2MEN1KMT2A
Hydrochloric Acid SCHEMBL7537987 0.81 GRM1 (0.72) EGFRGRM1ERBB2MEN1KMT2A
SCHEMBL7534837 0.80 EGFR (0.67) EGFRGRM1ERBB2HDAC1HDAC6
SCHEMBL11902821 0.78 EGFR (0.70) EGFRGRM1ERBB2MEN1KMT2A
SCHEMBL868343 0.77 EGFR (0.69) EGFRGRM1ERBB2MEN1KMT2A
Hydrochloric Acid SCHEMBL7541622 0.76 LMNA (0.52) EGFRLMNAMAPTHTTSMN1; SMN2
SCHEMBL16994115 0.75 EGFR (0.64) EGFRERBB2ERBB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1141298-A Pyrimidine-fused heterocyclic compound anti-cancer agents PFIZER (US) 1997-01-29 CN claimed
CN-1141298-A Pyrimidine-fused heterocyclic compound anti-cancer agents PFIZER (US) 1997-01-29 CN disclosed