SCHEMBL27460413

SCHEMBL27460413

[CH2]Oc1ccc(CCNC[C@H](O)COc2ccc(O[Si](C)(C)C(C)(C)C)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 13/20 0.58
ADRB1 P08588 8/20 0.58
ADRB2 P07550 7/20 0.58
KMT2A Q03164 3/20 0.50
ALDH1A1 P00352 1/20 0.50
MEN1 O00255 2/20 0.49
KCNH2 Q12809 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8587031 0.80 ADRB3 (0.50) ADRB3ADRB1ADRB2
SCHEMBL8587028 0.80 ADRB3 (0.50) ADRB3ADRB1ADRB2
SCHEMBL8794361 0.79 ADRB3 (0.46) ADRB3ADRB1ADRB2KMT2AALDH1A1
SCHEMBL24307676 0.73 ADRB3 (0.37) ADRB3ADRB1ADRB2KMT2AALDH1A1
SCHEMBL15275450 0.73 ADRB3 (0.76) ADRB3ADRB1ADRB2KMT2AMEN1
SCHEMBL9683368 0.71 ADRB3 (0.74) ADRB3ADRB1ADRB2KMT2AMEN1
SCHEMBL9683373 0.71 ADRB3 (0.74) ADRB3ADRB1ADRB2KMT2AMEN1
SCHEMBL7116296 0.71 ADRB3 (0.79) ADRB3ADRB1ADRB2KMT2AALDH1A1
SCHEMBL15445682 0.71 KMT2A (0.71) ADRB3ADRB1ADRB2KMT2AMEN1
SCHEMBL30206978 0.71 PREP (0.41) ADRB3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1159797-A Aryloxy and arylthiopropanolamine derivative suseful as beta 3-adrenoreceptor agonists and antagonists of the beta 1 and beta 2-adrenoreceptors and pharmaceutical composition thereof SMITHKLINE BEECHAM PLC (GB) 1997-09-17 CN disclosed