SCHEMBL27463129

SCHEMBL27463129

C[CH]c1c(C)cccc1-c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
PDCD1 Q15116 1/20 0.41
CD274 Q9NZQ7 1/20 0.41
CYP2A6 P11509 2/20 0.41
CYP2B6 P20813 1/20 0.41
ALDH1A1 P00352 5/20 0.39
HPGD P15428 2/20 0.39
TSHR P16473 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
PTGS2 P35354 1/20 0.38
ESR2 Q92731 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6548166 0.84 KDM4E (0.40) KDM4EPDCD1CD274CYP2A6CYP2B6
SCHEMBL309416 0.82 KDM4E (0.45) KDM4EPDCD1CD274CYP2A6CYP2B6
SCHEMBL1588208 0.82 KDM4E (0.41) KDM4EPDCD1CD274CYP2A6CYP2B6
SCHEMBL30404870 0.82 KDM4E (0.45) KDM4EPDCD1CD274CYP2A6CYP2B6
SCHEMBL27884523 0.77 KDM4E (0.41) KDM4EPDCD1CD274CYP2A6CYP2B6
SCHEMBL1610471 0.77 CYP2A6 (0.45) CYP2A6ALDH1A1TSHRCA1CA2
SCHEMBL30612770 0.74 CA12 (0.54) KDM4EPDCD1CD274CYP2A6CYP2B6
SCHEMBL29706107 0.74 ESR2 (0.54) KDM4EPDCD1CD274CYP2A6CYP2B6
SCHEMBL616 0.74 ESR2 (0.54) KDM4EPDCD1CD274CYP2A6CYP2B6
SCHEMBL7912257 0.73 NR1H2 (0.45) KDM4EPDCD1CD274ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1158269-C 4-aminothiazole derivs, their preparation and their use as inhibitors of cyclin-dependent kinases ������ҩ�����޹�˾ 2004-07-21 CN disclosed
CN-1276789-A 4-aminothiazole derivatives, their preparation and their use as inhibitors of cyclin dependent kinases AGOURON PHARMA (US) 2000-12-13 CN disclosed