SCHEMBL27477249

SCHEMBL27477249

CC=CCn1c(C)c(C)c2cnnc(C=Cc3ccccc3)c21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.34
GRM4 Q14833 2/20 0.33
HTR2A P28223 3/20 0.33
SIGMAR1 Q99720 3/20 0.33
CHRM2 P08172 2/20 0.33
CHRM4 P08173 2/20 0.33
CHRM5 P08912 2/20 0.33
ADRA2A P08913 2/20 0.33
CHRM1 P11229 2/20 0.33
ADRB3 P13945 2/20 0.33
ADRA2C P18825 2/20 0.33
CHRM3 P20309 2/20 0.33
S1PR1 P21453 2/20 0.33
FPR1 P21462 2/20 0.33
SLC6A2 P23975 2/20 0.33
HRH2 P25021 2/20 0.33
FPR3 P25089 2/20 0.33
AGTR1 P30556 2/20 0.33
GPR183 P32249 2/20 0.33
OPRM1 P35372 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27477248 1.00 NPSR1 (0.34) NPSR1GRM4HTR2ASIGMAR1CHRM2
SCHEMBL27477680 0.87 MEN1 (0.41) GRM4GPR35LMNATSHRKDM4E
SCHEMBL27501641 0.81 CYP1A2 (0.37) GRM4HTR2ASIGMAR1LMNAHTR2C
SCHEMBL27478116 0.79 CYP1A2 (0.51) GRM4GRM5
SCHEMBL7476839 0.79 NPSR1 (0.40) NPSR1HTR2ASIGMAR1CHRM2CHRM4
SCHEMBL7478191 0.77 ALDH1A1 (0.34) NPSR1LMNATSHRKDM4EALDH1A1
SCHEMBL7478196 0.77 ALDH1A1 (0.34) NPSR1LMNATSHRKDM4EALDH1A1
SCHEMBL7481101 0.75 CYP1A2 (0.52) NPSR1LMNATSHRALDH1A1MAPK1
SCHEMBL7481098 0.75 CYP1A2 (0.52) NPSR1LMNATSHRALDH1A1MAPK1
SCHEMBL7479782 0.75 CYP1A2 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1143964-A Pyrrolopyridazine derivative SANKYO CO (JP) 1997-02-26 CN claimed
CN-1143964-A Pyrrolopyridazine derivative SANKYO CO (JP) 1997-02-26 CN disclosed