SCHEMBL27486255

SCHEMBL27486255

Cc1cccc(NCc2ccncc2)c1C(=O)Nc1ccc(CN)cc1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 1/20 0.51
TYK2 P29597 1/20 0.51
FLT1 P17948 13/20 0.51
NAMPT P43490 2/20 0.50
LMNA P02545 1/20 0.49
KDR P35968 13/20 0.48
ABL1 P00519 1/20 0.45
EGFR P00533 1/20 0.45
CSF1R P07333 1/20 0.45
PDGFRB P09619 1/20 0.45
KIT P10721 1/20 0.45
FLT4 P35916 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4974383 0.91 KDR (0.58) ADRA2CTYK2FLT1NAMPTLMNA
SCHEMBL4976745 0.89 KDR (0.59) ADRA2CTYK2FLT1NAMPTLMNA
SCHEMBL27467101 0.82 KDR (0.67) FLT1KDRABL1EGFRCSF1R
SCHEMBL1715510 0.79 ADRA2C (0.63) ADRA2CNAMPT
SCHEMBL4978331 0.77 KDR (0.61) TYK2FLT1NAMPTKDR
SCHEMBL1715367 0.76 ADRA2C (0.53) ADRA2CFLT1NAMPT
SCHEMBL27554072 0.75 PLG (0.50) TYK2
SCHEMBL4979677 0.74 KDR (0.71) ADRA2CTYK2FLT1NAMPTKDR
SCHEMBL27485937 0.73 KDR (0.70) FLT1KDRABL1EGFRCSF1R
SCHEMBL27824623 0.72 PLG (0.47) TYK2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1152014-C N-aryl (thio) anthranilic acid amide derivatives, their prepn. and their use as VEGF receptor tyrosine kinase inhibitors ��˹��ŵ�� 2004-06-02 CN claimed
CN-1331680-A N-aryl (thio) anthranilic acid amide derivatives, their prepn. and their use as VEGF receptor tyrosine kinase inhibitors NOVARTIS AG (CH) 2002-01-16 CN claimed
CN-1152014-C N-aryl (thio) anthranilic acid amide derivatives, their prepn. and their use as VEGF receptor tyrosine kinase inhibitors ��˹��ŵ�� 2004-06-02 CN disclosed
CN-1331680-A N-aryl (thio) anthranilic acid amide derivatives, their prepn. and their use as VEGF receptor tyrosine kinase inhibitors NOVARTIS AG (CH) 2002-01-16 CN disclosed